Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50000682
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50261110BDBM50261110(Ethyl [(3aR,4aR,8aR,9aS)-9(S)-[(E)-2-[5-(3-fluorop...)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at PAR1 in human platelet-rich plasma assessed as reduction in TRAP-stimulated platelet aggregation preincubated for 20 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50261110BDBM50261110(Ethyl [(3aR,4aR,8aR,9aS)-9(S)-[(E)-2-[5-(3-fluorop...)
Affinity DataIC50: 64nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50261110BDBM50261110(Ethyl [(3aR,4aR,8aR,9aS)-9(S)-[(E)-2-[5-(3-fluorop...)
Affinity DataIC50: 81nMAssay Description:Antagonist activity at PAR1 in human platelet-rich plasma assessed as reduction in thrombin-stimulated platelet aggregation preincubated for 3 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257953BDBM50257953(CHEMBL4101591)
Affinity DataIC50: 650nMAssay Description:Antagonist activity at PAR1 in human platelet-rich plasma assessed as reduction in thrombin-stimulated platelet aggregation preincubated for 3 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257953BDBM50257953(CHEMBL4101591)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258055BDBM50258055(CHEMBL4084812)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257953BDBM50257953(CHEMBL4101591)
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at PAR1 in human platelet-rich plasma assessed as reduction in TRAP-stimulated platelet aggregation preincubated for 20 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258008BDBM50258008(CHEMBL4069403)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258033BDBM50258033(CHEMBL4077763)
Affinity DataIC50: 7.00E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258034BDBM50258034(CHEMBL4091623)
Affinity DataIC50: 8.10E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258011BDBM50258011(CHEMBL4065905)
Affinity DataIC50: 8.70E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258025BDBM50258025(CHEMBL4101239)
Affinity DataIC50: 9.10E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258026BDBM50258026(CHEMBL4065873)
Affinity DataIC50: 9.50E+3nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257976BDBM50257976(CHEMBL4092540)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258031BDBM50258031(CHEMBL4069486)
Affinity DataIC50: 1.20E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257975BDBM50257975(CHEMBL4093491)
Affinity DataIC50: 1.40E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258013BDBM50258013(CHEMBL4062114)
Affinity DataIC50: 1.40E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258021BDBM50258021(CHEMBL4100310)
Affinity DataIC50: 1.70E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258027BDBM50258027(CHEMBL4071756)
Affinity DataIC50: 1.90E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257983BDBM50257983(CHEMBL4072202)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257984BDBM50257984(CHEMBL4092965)
Affinity DataIC50: 2.10E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258017BDBM50258017(CHEMBL4083850)
Affinity DataIC50: 2.30E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258009BDBM50258009(CHEMBL4095795)
Affinity DataIC50: 2.90E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257972BDBM50257972(CHEMBL4066290)
Affinity DataIC50: 3.20E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258032BDBM50258032(CHEMBL4088070)
Affinity DataIC50: 5.50E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257971BDBM50257971(CHEMBL4074902)
Affinity DataIC50: 8.70E+4nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258024BDBM50258024(CHEMBL4074508)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257940BDBM50257940(CHEMBL4064870)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257978BDBM50257978(CHEMBL4104074)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258023BDBM50258023(CHEMBL4077889)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257977BDBM50257977(CHEMBL4086167)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258022BDBM50258022(CHEMBL4092571)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258029BDBM50258029(CHEMBL4085223)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257982BDBM50257982(CHEMBL4063603)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257981BDBM50257981(CHEMBL4074969)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258028BDBM50258028(CHEMBL4066363)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257952BDBM50257952(CHEMBL4102764)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257980BDBM50257980(CHEMBL4101654)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257979BDBM50257979(CHEMBL4093927)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258059BDBM50258059(CHEMBL4078212)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257974BDBM50257974(CHEMBL4104026)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258058BDBM50258058(CHEMBL4093859)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257973BDBM50257973(CHEMBL4086105)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257999BDBM50257999(CHEMBL4104430)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257998BDBM50257998(CHEMBL4080194)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50257997BDBM50257997(CHEMBL4096709)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258035BDBM50258035(CHEMBL4073470)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258012BDBM50258012(CHEMBL4070740)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
Shandong University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258010BDBM50258010(CHEMBL4092762)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human PAR1 expressed in HEK293 cells co-expressing Galpha15 assessed as inhibition of haTRAP-induced calcium mobilization prei...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2019
Entry Details Article
PubMed