Compile Data Set for Download or QSAR
Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 50002164
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454441BDBM50454441(CHEMBL4217448)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454379BDBM50454379(CHEMBL4205123)
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454411BDBM50454411(CHEMBL4209151)
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454402BDBM50454402(CHEMBL4209357)
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454399BDBM50454399(CHEMBL4215419)
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454410BDBM50454410(CHEMBL4212641)
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454392BDBM50454392(CHEMBL4204526)
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454382BDBM50454382(CHEMBL4206688)
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454396BDBM50454396(CHEMBL4207754)
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454384BDBM50454384(CHEMBL4205779)
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454453BDBM50454453(CHEMBL4211020)
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454397BDBM50454397(CHEMBL4215514)
Affinity DataIC50: 3nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50139171BDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 4nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454383BDBM50454383(CHEMBL4206359)
Affinity DataIC50: 4nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454387BDBM50454387(CHEMBL4216304)
Affinity DataIC50: 4nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454386BDBM50454386(CHEMBL4205084)
Affinity DataIC50: 5nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454404BDBM50454404(CHEMBL4209987)
Affinity DataIC50: 5nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454385BDBM50454385(CHEMBL4218213)
Affinity DataIC50: 6nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454456BDBM50454456(CHEMBL4213505)
Affinity DataIC50: 6nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454393BDBM50454393(CHEMBL4216190)
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454395BDBM50454395(CHEMBL4203989)
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454440BDBM50454440(CHEMBL4217685)
Affinity DataIC50: 9nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454445BDBM50454445(CHEMBL4203392)
Affinity DataIC50: 9nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454457BDBM50454457(CHEMBL4203224)
Affinity DataIC50: 9nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454403BDBM50454403(CHEMBL4210799)
Affinity DataIC50: 10nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454389BDBM50454389(CHEMBL4216726)
Affinity DataIC50: 11nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454401BDBM50454401(CHEMBL4202527)
Affinity DataIC50: 12nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454394BDBM50454394(CHEMBL4205921)
Affinity DataIC50: 12nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454390BDBM50454390(CHEMBL4215592)
Affinity DataIC50: 13nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454449BDBM50454449(CHEMBL4211337)
Affinity DataIC50: 14nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454391BDBM50454391(CHEMBL4204994)
Affinity DataIC50: 17nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454380BDBM50454380(CHEMBL4216857)
Affinity DataIC50: 21nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454381BDBM50454381(CHEMBL4216734)
Affinity DataIC50: 25nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454442BDBM50454442(CHEMBL4204402)
Affinity DataIC50: 33nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454446BDBM50454446(CHEMBL4209469)
Affinity DataIC50: 40nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454444BDBM50454444(CHEMBL4208684)
Affinity DataIC50: 49nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454443BDBM50454443(CHEMBL4204120)
Affinity DataIC50: 50nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454388BDBM50454388(CHEMBL4218452)
Affinity DataIC50: 55nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454398BDBM50454398(CHEMBL4203836)
Affinity DataIC50: 66nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454454BDBM50454454(CHEMBL4209102)
Affinity DataIC50: 122nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454439BDBM50454439(CHEMBL4206205)
Affinity DataIC50: 135nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454400BDBM50454400(CHEMBL4216039)
Affinity DataIC50: 210nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454447BDBM50454447(CHEMBL4215880)
Affinity DataIC50: 378nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454428BDBM50454428(CHEMBL4211689)
Affinity DataIC50: 458nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454455BDBM50454455(CHEMBL4206833)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454379BDBM50454379(CHEMBL4205123)
Affinity DataIC50: 5.91E+3nMAssay Description:Inhibition of human PLK1 kinase domain using 5-TAMRA-RGSFNDTLDFD-NH2 substrate and ATP incubated for 90 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454411BDBM50454411(CHEMBL4209151)
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of human PLK1 kinase domain using 5-TAMRA-RGSFNDTLDFD-NH2 substrate and ATP incubated for 90 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454453BDBM50454453(CHEMBL4211020)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of human PLK1 kinase domain using 5-TAMRA-RGSFNDTLDFD-NH2 substrate and ATP incubated for 90 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454396BDBM50454396(CHEMBL4207754)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of human PLK1 kinase domain using 5-TAMRA-RGSFNDTLDFD-NH2 substrate and ATP incubated for 90 mins by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Semmelweis University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454452BDBM50454452(CHEMBL4212016)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
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