Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50005450
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492205BDBM50492205(CHEMBL2397859)
Affinity DataIC50: 111nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492198BDBM50492198(CHEMBL2397840)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492209BDBM50492209(CHEMBL2397838)
Affinity DataIC50: 199nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492197BDBM50492197(CHEMBL2397841)
Affinity DataIC50: 247nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492204BDBM50492204(CHEMBL2397839)
Affinity DataIC50: 249nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492196BDBM50492196(CHEMBL2397850)
Affinity DataIC50: 309nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492195BDBM50492195(CHEMBL2397858)
Affinity DataIC50: 342nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492200BDBM50492200(CHEMBL2397849)
Affinity DataIC50: 354nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492194BDBM50492194(CHEMBL2397857)
Affinity DataIC50: 520nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492201BDBM50492201(CHEMBL2397851)
Affinity DataIC50: 607nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492199BDBM50492199(CHEMBL2397853)
Affinity DataIC50: 641nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492203BDBM50492203(CHEMBL2397852)
Affinity DataIC50: 774nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492193BDBM50492193(CHEMBL2397860)
Affinity DataIC50: 818nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492192BDBM50492192(CHEMBL2397854)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492202BDBM50492202(CHEMBL2397847)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492191BDBM50492191(CHEMBL2397855)
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492190BDBM50492190(CHEMBL2397846)
Affinity DataIC50: 7.01E+3nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492207BDBM50492207(CHEMBL2397845)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492208BDBM50492208(CHEMBL2397856)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492188BDBM50492188(CHEMBL2397843)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492187BDBM50492187(CHEMBL2397848)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492206BDBM50492206(CHEMBL2397844)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Jeil Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50492189BDBM50492189(CHEMBL2397842)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human GSK3 using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by [33P-gamma]-ATP addition m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed