Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50008633
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521018BDBM50521018(LG-190178)
Affinity DataEC50:  7.70nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50200182BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  100nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521014BDBM50521014(CHEMBL4459512)
Affinity DataEC50:  100nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521012BDBM50521012(CHEMBL4522782)
Affinity DataEC50:  400nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521017BDBM50521017(CHEMBL4524451)
Affinity DataEC50:  600nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521015BDBM50521015(CHEMBL4580825)
Affinity DataEC50:  600nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521013BDBM50521013(CHEBI:17933 | Calcifediol)
Affinity DataEC50:  600nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521020BDBM50521020(CHEMBL4459996)
Affinity DataEC50:  700nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50030475BDBM50030475(CHEBI:28940 | 7-Dehydrocholesterol | Cholecalcifer...)
Affinity DataEC50:  900nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521019BDBM50521019(CHEMBL4449816)
Affinity DataEC50:  1.30E+3nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521021BDBM50521021(CHEMBL4439766)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
University of Connecticut

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50521016BDBM50521016(CHEMBL4438180)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of VDR in mouse ASZ001 cells assessed as change in Cyp24A1 mRNA expression after 48 hrs by q-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed