Found 9 Enz. Inhib. hit(s) with all data for entry = 50010414 TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Ocean University Of China
Curated by ChEMBL
Ocean University Of China
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: 5.57E+3nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using isoform-specific probe substrates incubated for 15 to 30 mins by by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of CYP2C19 in human liver microsomes using isoform-specific probe substrates incubated for 15 to 30 mins by by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.93E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomes using isoform-specific probe substrates incubated for 15 to 30 mins by by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Ocean University Of China
Curated by ChEMBL
Ocean University Of China
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: 3.93E+4nMAssay Description:Inhibition of CYP2B6 in human liver microsomes using isoform-specific probe substrates incubated for 15 to 30 mins by by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5.41E+4nMAssay Description:Inhibition of CYP2C8 in human liver microsomes using isoform-specific probe substrates incubated for 15 to 30 mins by by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using isoform-specific probe substrates incubated for 15 to 30 mins by by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using isoform-specific probe substrates incubated for 15 to 30 mins by by LC-MS/MS analysisMore data for this Ligand-Target Pair
