Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50011271
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104439BDBM50104439(4-{2-Oxo-3-[4-(4-phenyl-butylsulfanyl)-phenoxy]-pr...)
Affinity DataIC50: 240nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104445BDBM50104445(1-[2-(4-Carboxy-2-fluoro-phenoxy)-ethyl]-3-dodecan...)
Affinity DataIC50: 440nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104453BDBM50104453(1-[2-(4-Carboxy-2-chloro-phenoxy)-ethyl]-3-dodecan...)
Affinity DataIC50: 520nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104444BDBM50104444(1-[2-(4-Carboxy-2-methyl-phenoxy)-ethyl]-3-dodecan...)
Affinity DataIC50: 570nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104456BDBM50104456(1-[2-(4-Carboxy-2,6-difluoro-phenoxy)-ethyl]-3-dod...)
Affinity DataIC50: 640nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104443BDBM50104443(1-[4-(4-Carboxy-phenoxy)-butyl]-3-dodecanoyl-1H-in...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104441BDBM50104441(1-[2-(4-Carboxy-2,6-dichloro-phenoxy)-ethyl]-3-dod...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104455BDBM50104455(1-[3-(4-Carboxy-phenyl)-propyl]-3-dodecanoyl-1H-in...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104454BDBM50104454(1-[2-(4-Carboxy-3-hydroxy-phenoxy)-ethyl]-3-dodeca...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104452BDBM50104452(1-[2-(4-Carboxy-3-methoxy-phenoxy)-ethyl]-3-dodeca...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104446BDBM50104446(1-{2-[(4-Carboxy-phenyl)-methyl-amino]-ethyl}-3-do...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104451BDBM50104451(1-[2-(4-Carboxy-3-chloro-phenoxy)-ethyl]-3-dodecan...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104449BDBM50104449(1-[2-(4-Carboxy-2-nitro-phenoxy)-ethyl]-3-dodecano...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104442BDBM50104442(1-[3-(4-Carboxy-phenoxy)-propyl]-3-dodecanoyl-1H-i...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104438BDBM50104438(1-[2-(4-Carboxy-2,6-dimethyl-phenoxy)-ethyl]-3-dod...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104450BDBM50104450(1-[2-(4-Carboxy-2-methoxy-phenoxy)-ethyl]-3-dodeca...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104440BDBM50104440(1-[2-(4-Carboxy-2-hydroxy-phenoxy)-ethyl]-3-dodeca...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
University of MüNster

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104448BDBM50104448(1-[2-(4-Carboxy-phenylamino)-ethyl]-3-dodecanoyl-1...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of cytosolic phospholipase A2 by measuring the calcium ionophore A-23,187-induced arachidonic acid release from human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed