Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50011960
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50552663BDBM50552663(CHEMBL4746871)
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells using Biotin-H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50552663BDBM50552663(CHEMBL4746871)
Affinity DataKd:  2.69E+3nMAssay Description:Binding affinity to recombinant human N-terminal His6-tagged lysine dye- labeled 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50552663BDBM50552663(CHEMBL4746871)
Affinity DataKd:  2.70E+3nMAssay Description:Binding affinity to recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells by SPR a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50552664BDBM50552664(CHEMBL4740162)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells using Biotin-H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50552665BDBM50552665(CHEMBL4743203)
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells using Biotin-H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50552666BDBM50552666(CHEMBL4757490)
Affinity DataIC50: 1.78E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells using Biotin-H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50552670BDBM50552670(CHEMBL4746119)
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells using Biotin-H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50552667BDBM50552667(CHEMBL4798544)
Affinity DataIC50: 3.13E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells using Biotin-H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50552671BDBM50552671(CHEMBL4741661)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells using Biotin-H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50552669BDBM50552669(CHEMBL4753650)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells using Biotin-H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetTP53-binding protein 1(Human)
Yantai University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50552668BDBM50552668(CHEMBL4787042)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged 53BP1 TTD (1484 to1603 residues) expressed in Escherichia coli BL21 (DE3) cells using Biotin-H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed