Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50012240
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555811BDBM50555811(CHEMBL4745224)
Affinity DataIC50: 150nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555796BDBM50555796(CHEMBL3438703)
Affinity DataIC50: 560nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555816BDBM50555816(CHEMBL4760028)
Affinity DataIC50: 700nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555812BDBM50555812(CHEMBL4761539)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555807BDBM50555807(CHEMBL4777629)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555810BDBM50555810(CHEMBL4782777)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555793BDBM50555793(CHEMBL4797817)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555797BDBM50555797(CHEMBL3438700)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555814BDBM50555814(CHEMBL4791080)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555806BDBM50555806(CHEMBL3438738)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555798BDBM50555798(CHEMBL4762380)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555805BDBM50555805(CHEMBL4744278)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555808BDBM50555808(CHEMBL4761995)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555804BDBM50555804(CHEMBL4740225)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555803BDBM50555803(CHEMBL4745101)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555802BDBM50555802(CHEMBL4776067)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555801BDBM50555801(CHEMBL4741129)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555800BDBM50555800(CHEMBL4783486)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555799BDBM50555799(CHEMBL4751449)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555815BDBM50555815(CHEMBL4793574)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555813BDBM50555813(CHEMBL4744743)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555795BDBM50555795(CHEMBL3438720)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555794BDBM50555794(CHEMBL4748831)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555809BDBM50555809(CHEMBL4762190)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Chongqing University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50555792BDBM50555792(CHEMBL4794344)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of LDHA (unknown origin) in presence of NADH and sodium pyruvate measured after 10 mins by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed