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Found 14 Enz. Inhib. hit(s) with all data for entry = 50016554
TargetAndrogen receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50170576(1-(4-{1-[4-(2,3-Dihydroxy-propylamino)-3-methyl-ph...)
Affinity DataKi:  1.17E+3nMAssay Description:Binding affinity to androgen receptor by incubation with GST-hARLBD and [3H]-testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50170573(3-(4-{1-Ethyl-1-[4-(2-hydroxy-3,3-dimethyl-butoxy)...)
Affinity DataKi:  1.51E+3nMAssay Description:Binding affinity to androgen receptor by incubation with GST-hARLBD and [3H]-testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50170578(1-(4-{1-Ethyl-1-[4-(3-hydroxy-3-methyl-butylamino)...)
Affinity DataKi:  2.90E+3nMAssay Description:Binding affinity to androgen receptor by incubation with GST-hARLBD and [3H]-testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50170582(4-(4-{1-Ethyl-1-[4-(3-hydroxy-3-methyl-butylamino)...)
Affinity DataKi:  3.38E+3nMAssay Description:Binding affinity to androgen receptor by incubation with GST-hARLBD and [3H]-testosteroneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50170576(1-(4-{1-[4-(2,3-Dihydroxy-propylamino)-3-methyl-ph...)
Affinity DataIC50:  7.60nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50170573(3-(4-{1-Ethyl-1-[4-(2-hydroxy-3,3-dimethyl-butoxy)...)
Affinity DataIC50:  9nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50329704((R)-3-(4-(3-(4-((R)-2-hydroxy-3,3-dimethylbutoxy)-...)
Affinity DataIC50:  19nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50170578(1-(4-{1-Ethyl-1-[4-(3-hydroxy-3-methyl-butylamino)...)
Affinity DataIC50:  820nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50410422(CHEMBL199131)
Affinity DataIC50:  1.00E+3nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50410421(CHEMBL199122)
Affinity DataIC50:  1.00E+3nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50410423(CHEMBL198213)
Affinity DataIC50:  1.20E+3nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM36720(LG190155)
Affinity DataIC50:  1.90E+3nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50410420(CHEMBL198651)
Affinity DataIC50:  3.50E+3nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50170582(4-(4-{1-Ethyl-1-[4-(3-hydroxy-3-methyl-butylamino)...)
Affinity DataIC50:  6.80E+3nMAssay Description:Androgen antagonistic activity as inhibitory concentration against testosterone-induced SC-3 cell proliferationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed