Compile Data Set for Download or QSAR
Report error Found 67 Enz. Inhib. hit(s) with all data for entry = 50018604
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610205BDBM50610205(CHEMBL5268764)
Affinity DataKi:  0.300nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610205BDBM50610205(CHEMBL5268764)
Affinity DataKi:  0.400nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50144861BDBM50144861(3-(5-Methyl-isoxazol-3-yl)-6-(pyridin-2-ylmethoxy)...)
Affinity DataKi:  0.400nMAssay Description:Negative allosteric modulation of alpha1 GABAA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50144861BDBM50144861(3-(5-Methyl-isoxazol-3-yl)-6-(pyridin-2-ylmethoxy)...)
Affinity DataKi:  0.5nMAssay Description:Negative allosteric modulation of alpha5 GABAA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610197BDBM50610197(CHEMBL5283158)
Affinity DataKi:  1.70nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610218BDBM50610218(CHEMBL5279431)
Affinity DataKi:  2nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610197BDBM50610197(CHEMBL5283158)
Affinity DataKi:  3.60nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 133427BDBM133427(US8846719, 112)
Affinity DataKi:  4.40nMAssay Description:Negative allosteric modulation of alpha5 GABAA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610203BDBM50610203(CHEMBL5267248)
Affinity DataKi:  5.40nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610218BDBM50610218(CHEMBL5279431)
Affinity DataKi:  7nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610199BDBM50610199(CHEMBL5279584)
Affinity DataKi:  8nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610212BDBM50610212(CHEMBL5276178)
Affinity DataKi:  11nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610203BDBM50610203(CHEMBL5267248)
Affinity DataKi:  12nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610212BDBM50610212(CHEMBL5276178)
Affinity DataKi:  15nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610189BDBM50610189(CHEMBL5267241)
Affinity DataKi:  15nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610198BDBM50610198(CHEMBL5285179)
Affinity DataKi:  16nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610196BDBM50610196(CHEMBL5283624)
Affinity DataKi:  16nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610193BDBM50610193(CHEMBL5281879)
Affinity DataKi:  17nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610194BDBM50610194(CHEMBL5282000)
Affinity DataKi:  17nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610199BDBM50610199(CHEMBL5279584)
Affinity DataKi:  18nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610213BDBM50610213(CHEMBL5276982)
Affinity DataKi:  20nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610202BDBM50610202(CHEMBL5289385)
Affinity DataKi:  23nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610187BDBM50610187(CHEMBL5271002)
Affinity DataKi:  28nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610200BDBM50610200(CHEMBL5290343)
Affinity DataKi:  30nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610189BDBM50610189(CHEMBL5267241)
Affinity DataKi:  30nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610191BDBM50610191(CHEMBL5266848)
Affinity DataKi:  32nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610187BDBM50610187(CHEMBL5271002)
Affinity DataKi:  32nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610188BDBM50610188(CHEMBL5287850)
Affinity DataKi:  33nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610196BDBM50610196(CHEMBL5283624)
Affinity DataKi:  35nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610190BDBM50610190(CHEMBL5285035)
Affinity DataKi:  48nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610206BDBM50610206(CHEMBL5287391)
Affinity DataKi:  52nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610183BDBM50610183(CHEMBL5272593)
Affinity DataKi:  52nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610188BDBM50610188(CHEMBL5287850)
Affinity DataKi:  55nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610191BDBM50610191(CHEMBL5266848)
Affinity DataKi:  56nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610193BDBM50610193(CHEMBL5281879)
Affinity DataKi:  60nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610194BDBM50610194(CHEMBL5282000)
Affinity DataKi:  60nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610192BDBM50610192(CHEMBL5283694)
Affinity DataKi:  64nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610198BDBM50610198(CHEMBL5285179)
Affinity DataKi:  65nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610190BDBM50610190(CHEMBL5285035)
Affinity DataKi:  74nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610211BDBM50610211(CHEMBL5284313)
Affinity DataKi:  76nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610202BDBM50610202(CHEMBL5289385)
Affinity DataKi:  80nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610209BDBM50610209(CHEMBL5272704)
Affinity DataKi:  86nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610211BDBM50610211(CHEMBL5284313)
Affinity DataKi:  89nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610206BDBM50610206(CHEMBL5287391)
Affinity DataKi:  100nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610195BDBM50610195(CHEMBL5290905)
Affinity DataKi:  107nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610213BDBM50610213(CHEMBL5276982)
Affinity DataKi:  120nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610207BDBM50610207(CHEMBL5278670)
Affinity DataKi:  122nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610192BDBM50610192(CHEMBL5283694)
Affinity DataKi:  123nMAssay Description:Displacement of flumazenil from alpha1 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610183BDBM50610183(CHEMBL5272593)
Affinity DataKi:  132nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Gedeon Richter

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610215BDBM50610215(CHEMBL5275441)
Affinity DataKi:  138nMAssay Description:Displacement of flumazenil from alpha5 GABAA receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
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