Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50021538
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641838BDBM50641838(CHEMBL5568777)
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of full length human PDE10A incubated for 1 hr by topcount Scintillation plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641839BDBM50641839(CHEMBL5542796)
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of full length human PDE10A incubated for 1 hr by topcount Scintillation plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641835BDBM50641835(CHEMBL5542573)
Affinity DataIC50: 0.00300nMAssay Description:Inhibition of full length human PDE10A incubated for 1 hr by topcount Scintillation plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641834BDBM50641834(CHEMBL5572487)
Affinity DataIC50: 0.00300nMAssay Description:Inhibition of full length human PDE10A incubated for 1 hr by topcount Scintillation plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641837BDBM50641837(CHEMBL5562552)
Affinity DataIC50: 0.00400nMAssay Description:Inhibition of full length human PDE10A incubated for 1 hr by topcount Scintillation plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641836BDBM50641836(CHEMBL5589788)
Affinity DataIC50: 0.00400nMAssay Description:Inhibition of full length human PDE10A incubated for 1 hr by topcount Scintillation plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641840BDBM50641840(CHEMBL5590372)
Affinity DataIC50: 0.00900nMAssay Description:Inhibition of full length human PDE10A incubated for 1 hr by topcount Scintillation plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641833BDBM50641833(CHEMBL5564394)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641824BDBM50641824(CHEMBL5566865)
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641831BDBM50641831(CHEMBL5591146)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641828BDBM50641828(CHEMBL5592321)
Affinity DataIC50: 310nMAssay Description:Inhibition of recombinant PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641830BDBM50641830(CHEMBL5590916)
Affinity DataIC50: 314nMAssay Description:Inhibition of recombinant PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641826BDBM50641826(CHEMBL5571543)
Affinity DataIC50: 450nMAssay Description:Inhibition of recombinant PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641827BDBM50641827(CHEMBL5568853)
Affinity DataIC50: 730nMAssay Description:Inhibition of recombinant PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641825BDBM50641825(CHEMBL5569774)
Affinity DataIC50: 790nMAssay Description:Inhibition of recombinant PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641832BDBM50641832(CHEMBL5574496)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPyruvate kinase PKM(Human)
National Institute of Pharmaceutical Education and Research Ahmedabad (NIPER-A)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641829BDBM50641829(CHEMBL5593879)
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of recombinant PKM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed