Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50028876
TargetThromboxane A2 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50008805(S 145 | S-145,(+) | CHEMBL56941 | 7-(3-Benzenesulf...)
Affinity DataKd:  2.90nMAssay Description:Tested for binding affinity against platelet TXA2 receptor in washed human platelets using [125I]BOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane A2 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50279863((Z)-7-((1R,2S)-2-Benzenesulfonylamino-cyclopentyl)...)
Affinity DataKd:  7.5nMAssay Description:Tested for binding affinity against platelet TXA2 receptor in washed human platelets using [125I]BOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane A2 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50279864((Z)-7-((1R,2R)-2-Benzenesulfonylamino-cyclopentyl)...)
Affinity DataKd:  36nMAssay Description:Tested for binding affinity against platelet TXA2 receptor in washed human platelets using [125I]BOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane A2 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50279862((E)-9-Benzenesulfonylamino-non-5-enoic acid | CHEM...)
Affinity DataKd:  67nMAssay Description:Tested for binding affinity against platelet TXA2 receptor in washed human platelets using [125I]BOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane A2 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50008807(CHEMBL52003 | 9-Benzenesulfonylamino-nonanoic acid)
Affinity DataKd:  172nMAssay Description:Tested for binding affinity against platelet TXA2 receptor in washed human platelets using [125I]BOP as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article