Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50028876
TargetThromboxane A2 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50279862((E)-9-Benzenesulfonylamino-non-5-enoic acid | CHEM...)
Affinity DataKd:  67nMAssay Description:Tested for binding affinity against platelet TXA2 receptor in washed human platelets using [125I]-BOP as radioligandMore data for this Ligand-Target Pair
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TargetThromboxane A2 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50279863((Z)-7-((1R,2S)-2-Benzenesulfonylamino-cyclopentyl)...)
Affinity DataKd:  7.5nMAssay Description:Tested for binding affinity against platelet TXA2 receptor in washed human platelets using [125I]-BOP as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane A2 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50008807(9-Benzenesulfonylamino-nonanoic acid | CHEMBL52003)
Affinity DataKd:  172nMAssay Description:Tested for binding affinity against platelet TXA2 receptor in washed human platelets using [125I]-BOP as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane A2 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50279864((Z)-7-((1R,2R)-2-Benzenesulfonylamino-cyclopentyl)...)
Affinity DataKd:  36nMAssay Description:Tested for binding affinity against platelet TXA2 receptor in washed human platelets using [125I]-BOP as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane A2 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50008805(7-(3-Benzenesulfonylamino-bicyclo[2.2.1]hept-2-yl)...)
Affinity DataKd:  2.90nMAssay Description:Tested for binding affinity against platelet TXA2 receptor in washed human platelets using [125I]-BOP as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article