Compile Data Set for Download or QSAR
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Found 14 Enz. Inhib. hit(s) with all data for entry = 50028904
TargetProstaglandin G/H synthase 1/2(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM22971(2-[(2,6-dichloro-3-methylphenyl)amino]benzoic acid...)
Affinity DataIC50:  100nMAssay Description:Compound was evaluated in an intact RBL-1 cell line for inhibition of 5-CyclooxygenaseMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1/2(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280051(5-[2-(3-Trifluoromethyl-phenylamino)-pyridin-3-yl]...)
Affinity DataIC50:  190nMAssay Description:In vitro inhibitory activity against Cyclooxygenase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50048004(5-(2-(3-(trifluoromethyl)phenylamino)phenyl)-1,3,4...)
Affinity DataIC50:  270nMAssay Description:In vitro inhibitory activity against Cyclooxygenase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50048003(5-[2-(2,3-Dimethyl-phenylamino)-phenyl]-3H-[1,3,4]...)
Affinity DataIC50:  610nMAssay Description:In vitro inhibitory activity against Cyclooxygenase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50048007(5-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl]-3...)
Affinity DataIC50:  700nMAssay Description:Tested for inhibition of contractile effects of Tachykinin receptor 1 in guinea pig ileum preparation.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50048007(5-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl]-3...)
Affinity DataIC50:  740nMAssay Description:In vitro inhibitory activity of the compound against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50048004(5-(2-(3-(trifluoromethyl)phenylamino)phenyl)-1,3,4...)
Affinity DataIC50:  770nMAssay Description:In vitro inhibitory activity of the compound against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50047998(5-(2-(3-(trifluoromethyl)phenylamino)phenyl)-1,3,4...)
Affinity DataIC50:  850nMAssay Description:In vitro inhibitory activity against Cyclooxygenase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50047998(5-(2-(3-(trifluoromethyl)phenylamino)phenyl)-1,3,4...)
Affinity DataIC50:  870nMAssay Description:In vitro inhibitory activity of the compound against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280051(5-[2-(3-Trifluoromethyl-phenylamino)-pyridin-3-yl]...)
Affinity DataIC50:  990nMAssay Description:In vitro inhibitory activity of the compound against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50048003(5-[2-(2,3-Dimethyl-phenylamino)-phenyl]-3H-[1,3,4]...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50048009(5-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl]-3...)
Affinity DataIC50:  1.39E+3nMAssay Description:In vitro inhibitory activity of the compound against 5-lipoxygenase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50048009(5-[2-(2,6-Dichloro-3-methyl-phenylamino)-phenyl]-3...)
Affinity DataIC50:  1.75E+3nMAssay Description:In vitro inhibitory activity against Cyclooxygenase was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM22971(2-[(2,6-dichloro-3-methylphenyl)amino]benzoic acid...)
Affinity DataIC50:  2.40E+4nMAssay Description:Compound was evaluated in an intact RBL-1 cell line for inhibition of 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails Article