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Found 24 Enz. Inhib. hit(s) with all data for entry = 50029077
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281226(CHEMBL328736 | N-[(S)-1-[(2R,3S)-4-((R)-Butylsulfa...)
Affinity DataIC50:  0.350nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281231((S)-4-Methyl-2-[(S)-2-(2-methyl-propane-2-sulfonyl...)
Affinity DataIC50:  1.70nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281229(1H-Indole-2-carboxylic acid [(S)-1-[4-((S,S,R)-but...)
Affinity DataIC50:  11nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281234((S)-N-[(S)-4-((R,R)-Butylsulfamoyl)-1-cyclohexylme...)
Affinity DataIC50:  64nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281242((S)-N-[(S)-4-((R,R)-Butylsulfamoyl)-1-cyclohexylme...)
Affinity DataIC50:  240nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281233((S)-4-Methyl-2-(3-phenyl-propionylamino)-pentanoic...)
Affinity DataIC50:  3.50E+3nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281223((2S,3R,4S)-5-Cyclohexyl-2,3-dihydroxy-4-(4-methyl-...)
Affinity DataIC50:  1.40E+4nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281238((2S,3R,4S)-4-Amino-5-cyclohexyl-2,3-dihydroxy-pent...)
Affinity DataIC50:  1.40E+4nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281222((S)-N-[(S)-4-((S,R)-Butylsulfamoyl)-1-cyclohexylme...)
Affinity DataIC50:  2.10E+4nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281237(CHEMBL93724 | [(S)-1-((1S,2R,3S)-4-Butylsulfamoyl-...)
Affinity DataIC50:  5.20E+4nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281240((S)-N-[(S)-4-((S,R)-Butylsulfamoyl)-1-cyclohexylme...)
Affinity DataIC50:  1.40E+5nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281239((2R,3R,4S)-5-Cyclohexyl-2,3-dihydroxy-4-[3-(3H-imi...)
Affinity DataIC50:  3.10E+5nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281232((2R,3R,4S)-4-Amino-5-cyclohexyl-2,3-dihydroxy-pent...)
Affinity DataIC50:  4.70E+5nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281227((2R,3R,4S)-5-Cyclohexyl-2,3-dihydroxy-4-(4-methyl-...)
Affinity DataIC50:  6.80E+5nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281235(CHEMBL90415 | N-((1S,2R,3S)-4-Butylsulfamoyl-1-cyc...)
Affinity DataIC50: >1.00E+6nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281236((S)-2-Hydroxy-4-methyl-pentanoic acid ((1S,2R,3S)-...)
Affinity DataIC50: >1.00E+6nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281228(4-Methyl-pentanoic acid ((1S,2R,3S)-4-butylsulfamo...)
Affinity DataIC50: >1.00E+6nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281244((S)-2-Amino-N-[4-((S,R,R)-butylsulfamoyl)-1-cycloh...)
Affinity DataIC50: >1.00E+6nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281224(4-Methyl-pentanoic acid ((1S,2R,3R)-4-butylsulfamo...)
Affinity DataIC50: >1.00E+6nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281241(CHEMBL93587 | N-((1S,2R,3S)-4-Butylsulfamoyl-1-cyc...)
Affinity DataIC50: >1.00E+6nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281221(CHEMBL94013 | N-((1S,2R,3R)-4-Butylsulfamoyl-1-cyc...)
Affinity DataIC50: >1.00E+6nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281243((S)-2-Hydroxy-4-methyl-pentanoic acid ((1S,2R,3R)-...)
Affinity DataIC50: >1.00E+6nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281230(CHEMBL327891 | N-((1S,2R,3R)-4-Butylsulfamoyl-1-cy...)
Affinity DataIC50: >1.00E+6nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281225((S)-2-Amino-4-methyl-pentanoic acid [(2R,3S)-4-((R...)
Affinity DataIC50: >1.00E+6nMpH: 7.0Assay Description:The compound was tested for its inhibitory activity against human renal renin at pH 7More data for this Ligand-Target Pair
In DepthDetails Article