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Found 17 Enz. Inhib. hit(s) with all data for entry = 50029098
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281469(CHEMBL313955 | [3-Benzylcarbamoyl-3,3-difluoro-1-(...)
Affinity DataKi:  0.300nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281472((1-Benzyl-3-benzylcarbamoyl-3,3-difluoro-2-oxo-pro...)
Affinity DataKi:  0.600nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281466(CHEMBL86651 | [1-(1-Benzyl-3-benzylcarbamoyl-3,3-d...)
Affinity DataKi:  1nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281470(CHEMBL86924 | [1-Benzyl-3,3-difluoro-2-oxo-3-(trim...)
Affinity DataKi:  600nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281480(CHEMBL87473 | [1-Benzyl-3-(2,2-dimethyl-propylcarb...)
Affinity DataKi:  650nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281475((3-Benzylcarbamoyl-3,3-difluoro-2-oxo-1-trimethyls...)
Affinity DataKi:  2.50E+3nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281473((3-Benzylcarbamoyl-3,3-difluoro-2-oxo-1-trimethyls...)
Affinity DataKi:  1.20E+4nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281467(CHEMBL2370046 | {1-[1-(1-{1-Benzyl-3,3-difluoro-4-...)
Affinity DataKi:  1.60E+5nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281471(CHEMBL87633 | [(S)-1-(1-Benzyl-3-benzylcarbamoyl-3...)
Affinity DataKi:  4.00E+5nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281474(CHEMBL432761 | [1-Benzyl-3-(benzyl-methyl-carbamoy...)
Affinity DataKi:  5.00E+6nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281477((1-Benzyl-3,3-difluoro-2-oxo-4-phenylacetylamino-b...)
Affinity DataKi:  6.00E+7nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281464((1-Benzyl-3-benzylcarbamoyl-3,3-difluoro-2-oxo-pro...)
Affinity DataIC50:  4nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281476(CHEMBL224483 | [(S)-1-(1-Benzyl-3-benzylcarbamoyl-...)
Affinity DataIC50:  27nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281478(CHEMBL415082 | [1-(1-Benzyl-3,3-difluoro-2,4-dioxo...)
Affinity DataIC50:  100nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281468((1-Benzyl-3-carbamoyl-3,3-difluoro-2-oxo-propyl)-c...)
Affinity DataIC50:  3.00E+5nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281479(CHEMBL313819 | [1-(1-Benzyl-3-benzylcarbamoyl-3,3-...)
Affinity DataIC50:  7.50E+5nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50281465(CHEMBL315011 | [1-(1-Benzyl-3-benzylcarbamoyl-3,3-...)
Affinity DataIC50:  5.00E+6nMAssay Description:Tested for inhibitory activity against the recombinant HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails Article