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Found 18 Enz. Inhib. hit(s) with all data for entry = 50029134
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  0.290nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  2.30nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281671((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  10nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281671((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  10nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281673((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  53nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281674((S)-N-(1-Benzyl-2-phenyl-ethyl)-3-{(S)-2-[(S)-2-(2...)
Affinity DataIC50:  72nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281671((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  100nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281671((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  100nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281675((S)-3-{(S)-2-[(R)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  500nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281670((S)-3-{(S)-2-[(R)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  600nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281673((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  700nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281672((S)-N-(1-Benzyl-2-phenyl-ethyl)-3-{(S)-2-[(R)-2-(2...)
Affinity DataIC50:  700nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281675((S)-3-{(S)-2-[(R)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281676((S)-3-{(S)-2-[(R)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281676((S)-3-{(S)-2-[(R)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281670((S)-3-{(S)-2-[(R)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  2.20E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281674((S)-N-(1-Benzyl-2-phenyl-ethyl)-3-{(S)-2-[(S)-2-(2...)
Affinity DataIC50:  6.20E+3nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281672((S)-N-(1-Benzyl-2-phenyl-ethyl)-3-{(S)-2-[(R)-2-(2...)
Affinity DataIC50:  1.20E+4nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails Article