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Found 33 Enz. Inhib. hit(s) with all data for entry = 50029432
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284416(2-{[Acetyl-(3-octadecylcarbamoyloxymethyl-cyclobut...)
Affinity DataKi:  4.30nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284419(2-{[Acetyl-((2R,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataKi:  4.30nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284417(2-{[Acetyl-((2R,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataKi:  5.70nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataKi:  7.20nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284414(2-{[Acetyl-((2S,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataKi:  9.20nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284412(2-{[Acetyl-((2S,4S)-4-hexadecylcarbamoyloxymethyl-...)
Affinity DataKi:  9.80nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284420(2-{[Acetyl-((2S,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataKi:  9.80nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284414(2-{[Acetyl-((2S,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataKi:  15nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284422(2-{[Acetyl-((2S,4S)-4-hexadecyloxymethyl-oxetan-2-...)
Affinity DataKi:  15nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284423(2-{[Acetyl-((2R,4R)-4-hexadecyloxymethyl-thietan-2...)
Affinity DataKi:  20nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284413(2-{[Acetyl-((2S,4R)-4-hexadecyloxymethyl-oxetan-2-...)
Affinity DataKi:  21nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284415(1-Ethyl-2-{[((2R,4R)-4-hexadecylcarbamoyloxymethyl...)
Affinity DataKi:  26nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284410(1-Ethyl-2-{[(4-methoxy-benzoyl)-(4-octadecylcarbam...)
Affinity DataKi:  34nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284411(2-{[Acetyl-((2R,4R)-1-acetyl-4-octadecylcarbamoylo...)
Affinity DataKi:  35nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284421(1-Ethyl-2-{[((2S,4S)-4-hexadecyloxymethyl-thietan-...)
Affinity DataKi:  99nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284425(2-{[Acetyl-(1-benzoyl-4-octadecylcarbamoyloxymethy...)
Affinity DataKi:  104nMAssay Description:In vitro ability to displace [3H]-PAF from PAF receptor in rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284412(2-{[Acetyl-((2S,4S)-4-hexadecylcarbamoyloxymethyl-...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284411(2-{[Acetyl-((2R,4R)-1-acetyl-4-octadecylcarbamoylo...)
Affinity DataIC50:  29nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284423(2-{[Acetyl-((2R,4R)-4-hexadecyloxymethyl-thietan-2...)
Affinity DataIC50:  52nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)
Affinity DataIC50:  55nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284416(2-{[Acetyl-(3-octadecylcarbamoyloxymethyl-cyclobut...)
Affinity DataIC50:  56nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284419(2-{[Acetyl-((2R,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataIC50:  57nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284422(2-{[Acetyl-((2S,4S)-4-hexadecyloxymethyl-oxetan-2-...)
Affinity DataIC50:  57nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284417(2-{[Acetyl-((2R,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataIC50:  57nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284420(2-{[Acetyl-((2S,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataIC50:  61nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284415(1-Ethyl-2-{[((2R,4R)-4-hexadecylcarbamoyloxymethyl...)
Affinity DataIC50:  69nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284410(1-Ethyl-2-{[(4-methoxy-benzoyl)-(4-octadecylcarbam...)
Affinity DataIC50:  84nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284413(2-{[Acetyl-((2S,4R)-4-hexadecyloxymethyl-oxetan-2-...)
Affinity DataIC50:  95nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284414(2-{[Acetyl-((2S,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataIC50:  97nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284414(2-{[Acetyl-((2S,4R)-4-octadecylcarbamoyloxymethyl-...)
Affinity DataIC50:  101nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284421(1-Ethyl-2-{[((2S,4S)-4-hexadecyloxymethyl-thietan-...)
Affinity DataIC50:  119nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284425(2-{[Acetyl-(1-benzoyl-4-octadecylcarbamoyloxymethy...)
Affinity DataIC50:  138nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50251276(BN 52021 | CHEMBL514432 | GINKOLIDE B | Gingkolide...)
Affinity DataIC50:  418nMAssay Description:In vitro inhibitory activity against PAF-induced aggregation of rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails Article