Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50029446
TargetProlyl endopeptidase(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50284618BDBM50284618(4-(4-Formyl-thiazolidine-3-carbonyl)-thiazolidine-...)
Affinity DataIC50: 0.5nMAssay Description:Compound was evaluated for the inhibition of prolyl endopeptidase (PEP) purified from human peripheral blood mononuclear cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50284620BDBM50284620(2-(2-Dimethoxymethyl-pyrrolidine-1-carbonyl)-pyrro...)
Affinity DataIC50: 120nMAssay Description:Compound was evaluated for the inhibition of prolyl endopeptidase (PEP) purified from human peripheral blood mononuclear cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50284624BDBM50284624(2-(4-Dimethoxymethyl-thiazolidine-3-carbonyl)-pyrr...)
Affinity DataIC50: 350nMAssay Description:Compound was evaluated for the inhibition of prolyl endopeptidase (PEP) purified from human peripheral blood mononuclear cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50284617BDBM50284617(2-(2-[1,3]Dithiolan-2-yl-pyrrolidine-1-carbonyl)-p...)
Affinity DataIC50: 420nMAssay Description:Compound was evaluated for the inhibition of prolyl endopeptidase (PEP) purified from human peripheral blood mononuclear cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50038869BDBM50038869(2-(Pyrrolidine-1-carbonyl)-pyrrolidine-1-carboxyli...)
Affinity DataIC50: 600nMAssay Description:Compound was evaluated for the inhibition of prolyl endopeptidase (PEP) purified from human peripheral blood mononuclear cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50284619BDBM50284619(2-(2-[1,3]Dioxolan-2-yl-pyrrolidine-1-carbonyl)-py...)
Affinity DataIC50: 700nMAssay Description:Compound was evaluated for the inhibition of prolyl endopeptidase (PEP) purified from human peripheral blood mononuclear cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50284621BDBM50284621(4-(4-Dimethoxymethyl-thiazolidine-3-carbonyl)-thia...)
Affinity DataIC50: 2.60E+3nMAssay Description:Compound was evaluated for the inhibition of prolyl endopeptidase (PEP) purified from human peripheral blood mononuclear cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50284623BDBM50284623(2-[2-(4-Methoxymethyl-[1,3]dioxolan-2-yl)-pyrrolid...)
Affinity DataIC50: 6.50E+3nMAssay Description:Compound was evaluated for the inhibition of prolyl endopeptidase (PEP) purified from human peripheral blood mononuclear cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50284622BDBM50284622(2-(2-Hydroxymethyl-pyrrolidine-1-carbonyl)-pyrroli...)
Affinity DataIC50: 1.40E+4nMAssay Description:Compound was evaluated for the inhibition of prolyl endopeptidase (PEP) purified from human peripheral blood mononuclear cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article