Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50029475
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284885(4-methyl-14-(5-nitro-2-pyridyldisulfanyl)-12-oxa-4...)
Affinity DataIC50: 31nMAssay Description:Ability to displace [3H][D-Ala2,MePhe4,Gly-ol5]enkephalin ([3H]DAGO) from mu opioid receptors in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50450288(CHEMBL2112189)
Affinity DataIC50: 58nMAssay Description:Ability to displace [3H][D-Ala2,MePhe4,Gly-ol5]enkephalin ([3H]DAGO) from mu opioid receptors in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284885(4-methyl-14-(5-nitro-2-pyridyldisulfanyl)-12-oxa-4...)
Affinity DataEC50:  58nMAssay Description:Compound was evaluated for its binding affinity to mu opioid receptors in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50450288(CHEMBL2112189)
Affinity DataIC50: 68nMAssay Description:Ability to displace [3H][D-Ser2,Leu5]enkephalin-Thr ([3H]DSLET) from Opioid receptor delta 1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284885(4-methyl-14-(5-nitro-2-pyridyldisulfanyl)-12-oxa-4...)
Affinity DataIC50: 206nMAssay Description:Ability to displace [3H][D-Ser2,Leu5]enkephalin-Thr ([3H]DSLET) from Opioid receptor delta 1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284885(4-methyl-14-(5-nitro-2-pyridyldisulfanyl)-12-oxa-4...)
Affinity DataEC50:  402nMAssay Description:Compound was evaluated for its binding affinity to Opioid receptor delta 1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50450288(CHEMBL2112189)
Affinity DataEC50:  1.20E+3nMAssay Description:Compound was evaluated for its binding affinity to Opioid receptor delta 1 in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50450288(CHEMBL2112189)
Affinity DataEC50:  1.70E+3nMAssay Description:Ability to displace [3H][D-Ala2,MePhe4,Gly-ol5]enkephalin ([3H]DAGO) from mu opioid receptors in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article