Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50029600
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285986(2-[6-(4-Fluoro-phenyl)-3-(3-pyridin-3-yl-1H-pyrrol...)
Affinity DataKi:  0.700nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285993(6-(4-Fluoro-phenoxy)-3-(3-pyridin-3-yl-1H-pyrrolo[...)
Affinity DataKi:  1.70nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50035397(6-(4-Fluoro-phenyl)-3-((R)-3-pyridin-3-yl-1H-pyrro...)
Affinity DataKi:  3.80nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285994(CHEMBL98835 | [6-(4-Fluoro-phenyl)-1-(2-hydroxy-et...)
Affinity DataKi:  5nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286011(6-(4-Fluoro-phenyl)-3-(3-pyridin-3-yl-1H-pyrrolo[1...)
Affinity DataKi:  6nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286000(CHEMBL99583 | [6-(4-Fluoro-phenyl)-1-methyl-1H-ind...)
Affinity DataKi:  7nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285996(6-(4-Fluoro-phenyl)-3-(3-pyridin-3-yl-1H-pyrrolo[1...)
Affinity DataKi:  10nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286008(6-Pyridin-3-yl-3-(3-pyridin-3-yl-1H-pyrrolo[1,2-c]...)
Affinity DataKi:  11nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286009(6-Benzyl-3-(3-pyridin-3-yl-1H-pyrrolo[1,2-c]thiazo...)
Affinity DataKi:  13nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286001(6-Bromo-3-(3-pyridin-3-yl-1H-pyrrolo[1,2-c]thiazol...)
Affinity DataKi:  15nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285989(6-Benzyloxy-3-(3-pyridin-3-yl-1H-pyrrolo[1,2-c]thi...)
Affinity DataKi:  17nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285984(6-(4-Fluoro-phenylsulfanyl)-3-(3-pyridin-3-yl-1H-p...)
Affinity DataKi:  17nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285987(6-(4-Fluoro-phenyl)-3-(3-pyridin-3-yl-1H-pyrrolo[1...)
Affinity DataKi:  19nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286003(6-Phenyl-3-(3-pyridin-3-yl-1H-pyrrolo[1,2-c]thiazo...)
Affinity DataKi:  23nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285998(6-(4-Fluoro-phenyl)-3-(3-pyridin-3-yl-1H-pyrrolo[1...)
Affinity DataKi:  25nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286002(CHEMBL319325 | [1-(2-Amino-ethyl)-6-(4-fluoro-phen...)
Affinity DataKi:  38nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286004((1H-Indol-3-yl)-(3-pyridin-3-yl-1H-pyrrolo[1,2-c]t...)
Affinity DataKi:  53nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285995((6-Benzyloxy-1H-indol-3-yl)-(3-pyridin-3-yl-1H-pyr...)
Affinity DataKi:  64nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285988(CHEMBL98831 | [6-(4-Fluoro-phenyl)-1H-indol-3-yl]-...)
Affinity DataKi:  75nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285997(6-Chloro-3-(3-pyridin-3-yl-1H-pyrrolo[1,2-c]thiazo...)
Affinity DataKi:  89nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285991((7-Benzyloxy-1H-indol-3-yl)-(3-pyridin-3-yl-1H-pyr...)
Affinity DataKi:  90nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285985(3-(3-Pyridin-3-yl-1H-pyrrolo[1,2-c]thiazole-7-carb...)
Affinity DataKi:  95nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286006(3-(3-Pyridin-3-yl-1H-pyrrolo[1,2-c]thiazole-7-carb...)
Affinity DataKi:  110nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285990(5-Benzyloxy-3-(3-pyridin-3-yl-1H-pyrrolo[1,2-c]thi...)
Affinity DataKi:  120nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285983(3-[6-(4-Fluoro-phenyl)-3-(3-pyridin-3-yl-1H-pyrrol...)
Affinity DataKi:  160nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286010(7-Benzyloxy-3-(3-pyridin-3-yl-1H-pyrrolo[1,2-c]thi...)
Affinity DataKi:  170nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286005((5-Benzyloxy-1H-indol-3-yl)-(3-pyridin-3-yl-1H-pyr...)
Affinity DataKi:  180nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285999(CHEMBL98853 | Morpholin-4-yl-[3-(3-pyridin-3-yl-1H...)
Affinity DataKi:  225nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286007((4-Hydroxy-1H-indol-3-yl)-(3-pyridin-3-yl-1H-pyrro...)
Affinity DataKi:  327nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50285992(6-(4-Fluoro-phenyl)-3-(3-pyridin-3-yl-1H-pyrrolo[1...)
Affinity DataKi:  940nMAssay Description:Tested in vitro for antagonistic activity to displace [3H]-PAF from rabbit platelet membrane PAF receptorsMore data for this Ligand-Target Pair
In DepthDetails Article