Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50029607
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286106(Morphinan Cyclic Imine analogue | CHEMBL321570)
Affinity DataIC50: 0.150nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu opioid receptor in hartley guinea pig brain membrane in the presence of 100 nM of D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286104(Morphinan Cyclic Imine analogue | CHEMBL410909)
Affinity DataIC50: 0.25nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu opioid receptor in hartley guinea pig brain membrane in the presence of 100 nM of D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286106(Morphinan Cyclic Imine analogue | CHEMBL321570)
Affinity DataIC50: 0.260nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from Opioid receptor kappa 1 in hartley guinea pig brain membrane in the presence of 100 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286106(Morphinan Cyclic Imine analogue | CHEMBL321570)
Affinity DataIC50: 0.320nMAssay Description:Compound was tested for its ability to displace [3H]Cl-DPDPE from delta opioid receptor in hartley guinea pig brain membrane in the presence of 100 n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286103(Morphinan Cyclic Imine analogue | CHEMBL102092)
Affinity DataIC50: 0.330nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu opioid receptor in hartley guinea pig brain membrane in the presence of 100 nM of D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286105(Morphinan Cyclic Imine analogue | CHEMBL318636)
Affinity DataIC50: 0.360nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu opioid receptor in hartley guinea pig brain membrane in the presence of 100 nM of D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286103(Morphinan Cyclic Imine analogue | CHEMBL102092)
Affinity DataIC50: 0.520nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from Opioid receptor kappa 1 in hartley guinea pig brain membrane in the presence of 100 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286105(Morphinan Cyclic Imine analogue | CHEMBL318636)
Affinity DataIC50: 0.520nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from Opioid receptor kappa 1 in hartley guinea pig brain membrane in the presence of 100 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286101(Morphinan Cyclic Imine analogue | CHEMBL3037845)
Affinity DataIC50: 0.560nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu opioid receptor in hartley guinea pig brain membrane in the presence of 100 nM of D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286103(Morphinan Cyclic Imine analogue | CHEMBL102092)
Affinity DataIC50: 0.690nMAssay Description:Compound was tested for its ability to displace [3H]Cl-DPDPE from delta opioid receptor in hartley guinea pig brain membrane in the presence of 100 n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286105(Morphinan Cyclic Imine analogue | CHEMBL318636)
Affinity DataIC50: 0.710nMAssay Description:Compound was tested for its ability to displace [3H]Cl-DPDPE from delta opioid receptor in hartley guinea pig brain membrane in the presence of 100 n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286102(Morphinan Cyclic Imine analogue | CHEMBL353736)
Affinity DataIC50: 0.890nMAssay Description:Compound was tested for its ability to displace [3H]DAMGO from mu opioid receptor in hartley guinea pig brain membrane in the presence of 100 nM of D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286104(Morphinan Cyclic Imine analogue | CHEMBL410909)
Affinity DataIC50: 2.40nMAssay Description:Compound was tested for its ability to displace [3H]Cl-DPDPE from delta opioid receptor in hartley guinea pig brain membrane in the presence of 100 n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286106(Morphinan Cyclic Imine analogue | CHEMBL321570)
Affinity DataIC50: 2.60nMAssay Description:Compound was tested for its ability to displace bremazocine from Opioid receptor kappa 2 in hartley guinea pig brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286101(Morphinan Cyclic Imine analogue | CHEMBL3037845)
Affinity DataIC50: 4.70nMAssay Description:Compound was tested for its ability to displace bremazocine from Opioid receptor kappa 2 in hartley guinea pig brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286103(Morphinan Cyclic Imine analogue | CHEMBL102092)
Affinity DataIC50: 6.20nMAssay Description:Compound was tested for its ability to displace bremazocine from Opioid receptor kappa 2 in hartley guinea pig brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286105(Morphinan Cyclic Imine analogue | CHEMBL318636)
Affinity DataIC50: 9.20nMAssay Description:Compound was tested for its ability to displace bremazocine from Opioid receptor kappa 2 in hartley guinea pig brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286102(Morphinan Cyclic Imine analogue | CHEMBL353736)
Affinity DataIC50: 12nMAssay Description:Compound was tested for its ability to displace [3H]Cl-DPDPE from delta opioid receptor in hartley guinea pig brain membrane in the presence of 100 n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286104(Morphinan Cyclic Imine analogue | CHEMBL410909)
Affinity DataIC50: 17nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from Opioid receptor kappa 1 in hartley guinea pig brain membrane in the presence of 100 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286101(Morphinan Cyclic Imine analogue | CHEMBL3037845)
Affinity DataIC50: 34nMAssay Description:Compound was tested for its ability to displace [3H]Cl-DPDPE from delta opioid receptor in hartley guinea pig brain membrane in the presence of 100 n...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286102(Morphinan Cyclic Imine analogue | CHEMBL353736)
Affinity DataIC50: 97nMAssay Description:Compound was tested for its ability to displace [3H]U-69593 from Opioid receptor kappa 1 in hartley guinea pig brain membrane in the presence of 100 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286104(Morphinan Cyclic Imine analogue | CHEMBL410909)
Affinity DataIC50: 320nMAssay Description:Compound was tested for its ability to displace bremazocine from Opioid receptor kappa 2 in hartley guinea pig brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286102(Morphinan Cyclic Imine analogue | CHEMBL353736)
Affinity DataIC50: 331nMAssay Description:Compound was tested for its ability to displace bremazocine from Opioid receptor kappa 2 in hartley guinea pig brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50286101(Morphinan Cyclic Imine analogue | CHEMBL3037845)
Affinity DataIC50: 380nMAssay Description:Compound was tested for its ability to displace bremazocine from Opioid receptor kappa 2 in hartley guinea pig brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article