Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50029609
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50059319(1-[(R)-5-(3-Aza-bicyclo[3.2.2]non-3-yl)-1-methyl-2...)
Affinity DataIC50:  0.100nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286113(1-((2S,4R)-2-Methyl-6-phenyl-2,4-dihydro-1H-3,5,10...)
Affinity DataIC50:  1.80nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286121(1-[(R)-5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-...)
Affinity DataIC50:  2.70nMAssay Description:Compound was tested for its binding affinity against gastrin receptor in guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286119(1-(3-Ethyl-phenyl)-3-[5-(4-methyl-piperazin-1-yl)-...)
Affinity DataIC50:  4.90nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286121(1-[(R)-5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-...)
Affinity DataIC50:  7.60nMAssay Description:Compound was tested for its binding affinity by measuring the displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cor...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  8.5nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286118(1-[5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-2,3-...)
Affinity DataIC50:  9.80nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286120(1-[5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-2,3-...)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286112(1-[5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-2,3-...)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286115(1-(3-Methoxy-phenyl)-3-[5-(4-methyl-piperazin-1-yl...)
Affinity DataIC50:  31nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286116(1-[1-Methyl-5-(4-methyl-piperazin-1-yl)-2-oxo-2,3-...)
Affinity DataIC50:  121nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286122(1-[(S)-5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-...)
Affinity DataIC50:  270nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  736nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286117(1-(1-Methyl-2-oxo-5-piperazin-1-yl-2,3-dihydro-1H-...)
Affinity DataIC50:  880nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286113(1-((2S,4R)-2-Methyl-6-phenyl-2,4-dihydro-1H-3,5,10...)
Affinity DataIC50:  1.56E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50059319(1-[(R)-5-(3-Aza-bicyclo[3.2.2]non-3-yl)-1-methyl-2...)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286122(1-[(S)-5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-...)
Affinity DataIC50:  1.90E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286114(4-[1-Methyl-2-oxo-3-(3-m-tolyl-ureido)-2,3-dihydro...)
Affinity DataIC50: >3.00E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286117(1-(1-Methyl-2-oxo-5-piperazin-1-yl-2,3-dihydro-1H-...)
Affinity DataIC50: >3.00E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286115(1-(3-Methoxy-phenyl)-3-[5-(4-methyl-piperazin-1-yl...)
Affinity DataIC50: >3.00E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286121(1-[(R)-5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-...)
Affinity DataIC50: >3.00E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286119(1-(3-Ethyl-phenyl)-3-[5-(4-methyl-piperazin-1-yl)-...)
Affinity DataIC50: >3.00E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286114(4-[1-Methyl-2-oxo-3-(3-m-tolyl-ureido)-2,3-dihydro...)
Affinity DataIC50: >3.00E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286118(1-[5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-2,3-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286120(1-[5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-2,3-...)
Affinity DataIC50:  3.80E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286116(1-[1-Methyl-5-(4-methyl-piperazin-1-yl)-2-oxo-2,3-...)
Affinity DataIC50:  4.26E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50286112(1-[5-(4-Methyl-piperazin-1-yl)-2-oxo-1-propyl-2,3-...)
Affinity DataIC50:  5.31E+3nMAssay Description:Displacement of [125I]-BH CCK-8S from Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In DepthDetails Article