Compile Data Set for Download or QSAR
maximum 50k data
Found 66 Enz. Inhib. hit(s) with all data for entry = 50029613
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286172(CHEMBL320154 | Pyrrolidine-1-carboxylic acid (R)-3...)
Affinity DataIC50:  34nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286171(1-[(R)-1-(4-Benzoyl-piperidine-1-carbonyl)-4-oxo-4...)
Affinity DataIC50:  53nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286166(CHEMBL418987 | Pyrrolidine-1-carboxylic acid (R)-3...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286158(CHEMBL103312 | Phenyl-carbamic acid (R)-3-(4-benzo...)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286163(1-[(R)-3-Benzyloxy-2-(3-m-tolyl-ureido)-propionyl]...)
Affinity DataIC50:  160nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286148(1-[(S)-2-(4-Benzoyl-piperidin-1-yl)-2-oxo-1-phenyl...)
Affinity DataIC50:  170nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286177(CHEMBL104958 | Morpholine-4-carboxylic acid (R)-3-...)
Affinity DataIC50:  180nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286168(CHEMBL321072 | [(S)-1-[(S)-1-(4-Benzyl-piperidine-...)
Affinity DataIC50:  200nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286165(1-{1-((R)-Benzyloxymethyl)-2-[4-(4-fluoro-benzoyl)...)
Affinity DataIC50:  230nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286172(CHEMBL320154 | Pyrrolidine-1-carboxylic acid (R)-3...)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286158(CHEMBL103312 | Phenyl-carbamic acid (R)-3-(4-benzo...)
Affinity DataIC50:  290nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286150(1-[(R)-2-(4-Benzoyl-piperidin-1-yl)-1-benzyloxymet...)
Affinity DataIC50:  300nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286169(1-[(S)-2-(4-Benzoyl-piperidin-1-yl)-1-benzylsulfan...)
Affinity DataIC50:  390nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286156(4-(4-Benzoyl-piperidin-1-yl)-4-(R)-oxo-3-(3-m-toly...)
Affinity DataIC50:  410nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286165(1-{1-((R)-Benzyloxymethyl)-2-[4-(4-fluoro-benzoyl)...)
Affinity DataIC50:  420nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286157(1-{(R)-1-[(R)-(4-Benzoyl-piperidin-1-yl)-oxo-methy...)
Affinity DataIC50:  440nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286163(1-[(R)-3-Benzyloxy-2-(3-m-tolyl-ureido)-propionyl]...)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286174(CHEMBL320886 | [(S)-1-[(S)-1-(4-Benzoyl-piperidine...)
Affinity DataIC50:  640nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286159(5-(R)-Oxo-5-(4-phenylcarbamoyl-piperidin-1-yl)-4-(...)
Affinity DataIC50:  690nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286148(1-[(S)-2-(4-Benzoyl-piperidin-1-yl)-2-oxo-1-phenyl...)
Affinity DataIC50:  800nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286160(1-[(S)-2-(4-Benzoyl-piperidin-1-yl)-2-oxo-1-phenyl...)
Affinity DataIC50:  810nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286151((R)-5-(4-Benzoyl-piperidin-1-yl)-5-oxo-4-(3-m-toly...)
Affinity DataIC50:  900nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286151((R)-5-(4-Benzoyl-piperidin-1-yl)-5-oxo-4-(3-m-toly...)
Affinity DataIC50:  900nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286174(CHEMBL320886 | [(S)-1-[(S)-1-(4-Benzoyl-piperidine...)
Affinity DataIC50:  912nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286153(5-(4-Benzoylamino-piperidin-1-yl)-5-(R)-oxo-4-(3-m...)
Affinity DataIC50:  970nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286175(1-{1-[(R)-(4-Benzoyl-piperidin-1-yl)-oxo-methyl]-4...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286160(1-[(S)-2-(4-Benzoyl-piperidin-1-yl)-2-oxo-1-phenyl...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286156(4-(4-Benzoyl-piperidin-1-yl)-4-(R)-oxo-3-(3-m-toly...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286157(1-{(R)-1-[(R)-(4-Benzoyl-piperidin-1-yl)-oxo-methy...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286169(1-[(S)-2-(4-Benzoyl-piperidin-1-yl)-1-benzylsulfan...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286164(1-[(R)-2-(4-Acetyl-piperidin-1-yl)-1-benzyloxymeth...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286162(CHEMBL105303 | Dimethyl-carbamic acid (R)-3-(4-ben...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286166(CHEMBL418987 | Pyrrolidine-1-carboxylic acid (R)-3...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286176(1-[2-((R)-4-Benzoyl-piperidin-1-yl)-1-(1H-indol-3-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286177(CHEMBL104958 | Morpholine-4-carboxylic acid (R)-3-...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421364(CHEMBL2111654)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286162(CHEMBL105303 | Dimethyl-carbamic acid (R)-3-(4-ben...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286167(CHEMBL105618 | [2-(4-Benzoyl-piperidin-1-yl)-1-(1H...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286152((R)-5-(4-Benzoyl-piperidin-1-yl)-5-oxo-4-(3-m-toly...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286175(1-{1-[(R)-(4-Benzoyl-piperidin-1-yl)-oxo-methyl]-4...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286171(1-[(R)-1-(4-Benzoyl-piperidine-1-carbonyl)-4-oxo-4...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286170(1-[(R)-1-(4-Benzoyl-piperidine-1-carbonyl)-3-methy...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286159(5-(R)-Oxo-5-(4-phenylcarbamoyl-piperidin-1-yl)-4-(...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286152((R)-5-(4-Benzoyl-piperidin-1-yl)-5-oxo-4-(3-m-toly...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286154(CHEMBL101854 | [(S)-1-(4-Benzoyl-piperidine-1-carb...)
Affinity DataIC50: >2.10E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286149(1-[(R)-1-(4-Benzoyl-piperidine-1-carbonyl)-3-pheny...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286161(1-[(R)-3-Benzyloxy-2-(3-m-tolyl-ureido)-propionyl]...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286150(1-[(R)-2-(4-Benzoyl-piperidin-1-yl)-1-benzyloxymet...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50286173(1-[(R)-1-(4-Benzoyl-piperidine-1-carbonyl)-pentyl]...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKA receptor in guinea pig pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286167(CHEMBL105618 | [2-(4-Benzoyl-piperidin-1-yl)-1-(1H...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibitory activity towards binding of [125I]-Bolton-Hunter-CCK-8 to CCKB receptor in guinea pig cortical tissueMore data for this Ligand-Target Pair
In DepthDetails Article
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