Affinity DataIC50: 1.20nMAssay Description:Antagonistic activity against endothelin B (ETB) receptor using human girardi heart cells.More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonistic activity against endothelin A (ETA) receptor using human neuroblastoma cell line.More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+3nMAssay Description:Ability to block endothelin-1 (ET-1) stimulated arachidonic acid release in rabbit renal vascular smooth muscle cells (AARA) expressing recombinant r...More data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.10E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 9.50E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Ability to block sarafotoxin-6c (SRTX-6c) stimulated arachidonic acid release in chinese hamster ovary (CHO) cells expressing recombinant rat endothe...More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair