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Found 24 Enz. Inhib. hit(s) with all data for entry = 50029660
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286614(CHEMBL155943 | CHEMBL3143473 | Sodium; 2-[2-{2-[(2...)
Affinity DataIC50:  1.20nMAssay Description:Antagonistic activity against endothelin B (ETB) receptor using human girardi heart cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286622(Ac-W-F-F-N-Y-Y-W | CHEMBL405677)
Affinity DataIC50:  250nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286614(CHEMBL155943 | CHEMBL3143473 | Sodium; 2-[2-{2-[(2...)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonistic activity against endothelin A (ETA) receptor using human neuroblastoma cell line.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286619(Ac-bhg-F-N-Y-Y-W | CHEMBL385405)
Affinity DataIC50:  1.90E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286618(CHEMBL413880 | W-F-F-N--Y-Y-W)
Affinity DataIC50:  2.40E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286616(CHEMBL267610 | G-N-W-H-G-T-A-P-D-W-F-F-N-Y-Y-W)
Affinity DataIC50: >2.50E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286616(CHEMBL267610 | G-N-W-H-G-T-A-P-D-W-F-F-N-Y-Y-W)
Affinity DataIC50: >2.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286620(CHEMBL415614 | W-H-G-T-A-P-D-W-F-F-N-Y-Y-W)
Affinity DataIC50: >2.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286620(CHEMBL415614 | W-H-G-T-A-P-D-W-F-F-N-Y-Y-W)
Affinity DataIC50: >2.50E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286619(Ac-bhg-F-N-Y-Y-W | CHEMBL385405)
Affinity DataIC50:  4.30E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(CHEMBL413825 | Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His...)
Affinity DataIC50: >5.00E+3nMAssay Description:Ability to block endothelin-1 (ET-1) stimulated arachidonic acid release in rabbit renal vascular smooth muscle cells (AARA) expressing recombinant r...More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(CHEMBL413825 | Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His...)
Affinity DataIC50:  6.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(CHEMBL413825 | Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His...)
Affinity DataIC50:  6.50E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286622(Ac-W-F-F-N-Y-Y-W | CHEMBL405677)
Affinity DataIC50:  7.60E+3nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(CHEMBL413825 | Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His...)
Affinity DataIC50:  7.60E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(CHEMBL413825 | Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His...)
Affinity DataIC50:  7.80E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286615(Ac-w-F-F-N-Y-Y-W | CHEMBL441006)
Affinity DataIC50:  8.10E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286617(CHEMBL414917 | bhg-F-N-Y-Y-W)
Affinity DataIC50:  9.50E+3nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286617(CHEMBL414917 | bhg-F-N-Y-Y-W)
Affinity DataIC50:  1.30E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286615(Ac-w-F-F-N-Y-Y-W | CHEMBL441006)
Affinity DataIC50:  1.40E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286618(CHEMBL413880 | W-F-F-N--Y-Y-W)
Affinity DataIC50:  1.50E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286613(CHEMBL413825 | Cyclic (Gly1-Asp9) (Gly-Asn-Trp-His...)
Affinity DataIC50:  1.60E+4nMAssay Description:Ability to block sarafotoxin-6c (SRTX-6c) stimulated arachidonic acid release in chinese hamster ovary (CHO) cells expressing recombinant rat endothe...More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286621(CHEMBL264253 | F-F-N-Y-YW)
Affinity DataIC50: >2.50E+4nMAssay Description:Binding affinity in Chinese hamster ovary (CHO) cells stably transfected with human endothelin B (ETB) receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50286621(CHEMBL264253 | F-F-N-Y-YW)
Affinity DataIC50: >2.50E+4nMAssay Description:Binding affinity in LtK cells stably transfected with human endothelin A (ETA) receptorMore data for this Ligand-Target Pair
In DepthDetails Article