Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50029813
TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288232(2-[2-(carboxymethoxy)-4-(2-{4H,5H,6H,7H-thieno[2,3...)
Affinity DataIC50: 1.40nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288220((2-Carboxymethoxy-5-{2-[(4,5,6,7-tetrahydro-thieno...)
Affinity DataIC50: 4.70nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288220((2-Carboxymethoxy-5-{2-[(4,5,6,7-tetrahydro-thieno...)
Affinity DataIC50: 4.70nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288227((2-Carboxymethoxy-5-{2-[(5,6,7,8-tetrahydro-4H-thi...)
Affinity DataIC50: 6nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288218((2-Carboxymethoxy-5-{2-[(5,6,7,8-tetrahydro-4H-thi...)
Affinity DataIC50: 8.70nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288230((4-Carboxymethoxy-6-{2-[(4,5,6,7-tetrahydro-thieno...)
Affinity DataIC50: 9.80nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288229((2-Carboxymethoxy-5-{2-[(3-methyl-4,5,6,7-tetrahyd...)
Affinity DataIC50: 18nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288220((2-Carboxymethoxy-5-{2-[(4,5,6,7-tetrahydro-thieno...)
Affinity DataIC50: 28nMAssay Description:Inhibition of vWF binding to alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288225((4-{2-[(4,5,6,7-Tetrahydro-thieno[3,2-c]pyridine-2...)
Affinity DataIC50: 31nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288231({2-Carboxymethoxy-5-[2-(3-piperidin-4-yl-propionyl...)
Affinity DataIC50: 42nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288223(2-{4-[2-({3-benzyl-4H,5H,6H,7H-thieno[3,2-c]pyridi...)
Affinity DataIC50: 62nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50107402(2-[2-(2-Amino-5-guanidino-pentanoylamino)-acetylam...)
Affinity DataIC50: 76nMAssay Description:Inhibition of biotinylated fibrinogen binding to alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288224(3-(4-{2-[(4,5,6,7-Tetrahydro-thieno[3,2-c]pyridine...)
Affinity DataIC50: 80nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288233({2-Carboxymethoxy-5-[2-(2-piperidin-4-yl-acetylami...)
Affinity DataIC50: 100nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288226({2-Carboxymethoxy-5-[2-(4-piperidin-4-yl-butyrylam...)
Affinity DataIC50: 100nMAssay Description:Inhibition of biotinylated fibrinogen binding to alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288228((6-{2-[(4,5,6,7-Tetrahydro-thieno[3,2-c]pyridine-2...)
Affinity DataIC50: 100nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288219((2-Carboxymethoxy-4-{2-[(5,6-dihydro-4H-thieno[2,3...)
Affinity DataIC50: 100nMAssay Description:Inhibition of biotinylated fibrinogen binding to alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288234((5-Carboxymethoxy-2-{2-[(4,5,6,7-tetrahydro-thieno...)
Affinity DataIC50: 100nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288221((4-{2-[(4-Aminomethyl-cyclohexanecarbonyl)-amino]-...)
Affinity DataIC50: 730nMAssay Description:Inhibition of biotinylated fibrinogen binding to alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288222((3-Carboxymethoxy-5-{2-[(4,5,6,7-tetrahydro-thieno...)
Affinity DataIC50: 1.00E+3nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288235((2-Carboxymethoxy-4-{2-[(piperidine-4-carbonyl)-am...)
Affinity DataIC50: 1.00E+3nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50107402(2-[2-(2-Amino-5-guanidino-pentanoylamino)-acetylam...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of Vitronectin binding to GPIIb/IIIIa Vitronectin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50107402(2-[2-(2-Amino-5-guanidino-pentanoylamino)-acetylam...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of vWF binding to GPIIb/IIIIa receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetIntegrin alpha-IIb/beta-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50288220((2-Carboxymethoxy-5-{2-[(4,5,6,7-tetrahydro-thieno...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Vitronectin binding to GPIIb/IIIIa Vitronectin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article