Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for entry = 50029836
LigandPNGBDBM50288501(2-{2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta...)
Affinity DataIC50:  660nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288479(8-Chloro-11-(1-phenylmethanesulfonyl-piperidin-4-y...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288481(8-Chloro-11-(1-ethenesulfonyl-piperidin-4-ylidene)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288506(CHEMBL101603 | [(R)-2-[4-(8-Chloro-5,6-dihydro-ben...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288495(4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,2-b...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288498(8-Chloro-11-(1-methanesulfonyl-piperidin-4-ylidene...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288499(2-{2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288507(CHEMBL318268 | [(S)-2-[4-(8-Chloro-5,6-dihydro-ben...)
Affinity DataIC50:  3.05E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288502(2-[(R)-2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cycloh...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288478(2-{(R)-2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cycloh...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288480(2-{(R)-1-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cycloh...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288500(11-[1-(Butane-1-sulfonyl)-piperidin-4-ylidene]-8-c...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288505((R)-5-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohept...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288491(8-Chloro-11-(1-ethanesulfonyl-piperidin-4-ylidene)...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288509((S)-2-Amino-1-[4-(8-chloro-5,6-dihydro-benzo[5,6]c...)
Affinity DataIC50:  6.29E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288493(CHEMBL323298 | {2-[4-(8-Chloro-5,6-dihydro-benzo[5...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288490(1-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,...)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288504(CHEMBL101936 | N-{2-[4-(8-Chloro-5,6-dihydro-benzo...)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288497(CHEMBL432011 | {2-[4-(8-Chloro-5,6-dihydro-benzo[5...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288487(CHEMBL318886 | N-{2-[4-(8-Chloro-5,6-dihydro-benzo...)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288492(2-Benzylamino-1-[4-(8-chloro-5,6-dihydro-benzo[5,6...)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288489(2-{(R)-1-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cycloh...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288508(2-{(R)-1-Benzyl-2-[4-(8-chloro-5,6-dihydro-benzo[5...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288482(1-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288483(2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,...)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288486(2-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,...)
Affinity DataIC50: >1.10E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288488(1-[4-(8-Chloro-5,6-dihydro-benzo[5,6]cyclohepta[1,...)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288485(8-Chloro-11-[1-(octane-1-sulfonyl)-piperidin-4-yli...)
Affinity DataIC50: >1.20E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288484(8-Chloro-11-[1-(4-nitro-benzenesulfonyl)-piperidin...)
Affinity DataIC50: >1.20E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288494(8-Chloro-11-[1-(naphthalene-2-sulfonyl)-piperidin-...)
Affinity DataIC50: >1.20E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288496(8-Chloro-11-[1-(thiophene-2-sulfonyl)-piperidin-4-...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288503(2-Amino-1-[4-(8-chloro-5,6-dihydro-benzo[5,6]cyclo...)
Affinity DataIC50:  2.23E+4nMAssay Description:Inhibitory activity against protein farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails Article