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Found 24 Enz. Inhib. hit(s) with all data for entry = 50029904
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289172(CHEMBL367569 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289168(CHEMBL173643 | N-{4-Oxo-2-propyl-3-[2'-(2H-tetrazo...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289166(4'-[6-(3-Isopropyl-ureido)-4-oxo-2-propyl-4H-quina...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282471(CHEMBL168771 | N-[3-(2'-Benzoylsulfamoyl-biphenyl-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289170(CHEMBL408798 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289165(CHEMBL408799 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289163(CHEMBL368149 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289167(4'-[6-(3-Isopropyl-ureido)-4-oxo-2-propyl-4H-quina...)
Affinity DataIC50:  8.80nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289164(CHEMBL367095 | N-[3-(2'-Benzoylsulfamoyl-biphenyl-...)
Affinity DataIC50:  11nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282471(CHEMBL168771 | N-[3-(2'-Benzoylsulfamoyl-biphenyl-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289166(4'-[6-(3-Isopropyl-ureido)-4-oxo-2-propyl-4H-quina...)
Affinity DataIC50:  18nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289169(CHEMBL174080 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  20nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289171(CHEMBL172376 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  23nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289163(CHEMBL368149 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  24nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289169(CHEMBL174080 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  30nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289170(CHEMBL408798 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  49nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289165(CHEMBL408799 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  75nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289172(CHEMBL367569 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  200nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289164(CHEMBL367095 | N-[3-(2'-Benzoylsulfamoyl-biphenyl-...)
Affinity DataIC50:  350nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289167(4'-[6-(3-Isopropyl-ureido)-4-oxo-2-propyl-4H-quina...)
Affinity DataIC50:  630nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289168(CHEMBL173643 | N-{4-Oxo-2-propyl-3-[2'-(2H-tetrazo...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50289171(CHEMBL172376 | Macrocyclic Quinazolinone analogue)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to rat midbrain Angiotensin II receptor type 2More data for this Ligand-Target Pair
In DepthDetails Article