Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50029955
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289671((2S,4R)-6-Biphenyl-4-yl-2-butyl-4-[(S)-2-(4-methox...)
Affinity DataKi:  21nMAssay Description:Inhibition of Matrix metalloproteinase-3 by MCA peptide assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289668((2S,4R)-6-Biphenyl-4-yl-2-butyl-4-((S)-6-methylcar...)
Affinity DataKi:  42nMAssay Description:Inhibition of Matrix metalloproteinase-3 by MCA peptide assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289676((R)-2-[(S)-3-(Biphenyl-4-yloxy)-1-((S)-6-methylcar...)
Affinity DataKi:  77nMAssay Description:Inhibition of Matrix metalloproteinase-3 by MCA peptide assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289674((R)-2-[(S)-3-(4-Butyl-phenoxy)-1-((S)-6-methylcarb...)
Affinity DataKi:  550nMAssay Description:Inhibition of Matrix metalloproteinase-3 by MCA peptide assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289675((R)-2-[(S)-3-(4-Benzyl-phenoxy)-1-((S)-6-methylcar...)
Affinity DataKi:  552nMAssay Description:Inhibition of Matrix metalloproteinase-3 by MCA peptide assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289670((S)-2-[(R)-2-((S)-1-Hydroxycarbamoyl-ethyl)-4-meth...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Matrix metalloproteinase-3 by MCA peptide assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289673((2S,4R)-6-Biphenyl-4-yl-4-[(S)-2-(4-methoxy-phenyl...)
Affinity DataIC50:  81nMAssay Description:Inhibition of Matrix metalloproteinase-3 by MCA peptide assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289669((2S,4R)-4-[(S)-2-(4-Methoxy-phenyl)-1-methylcarbam...)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of Matrix metalloproteinase-3 by MCA peptide assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289667((R)-2-[(S)-3-(4-Cyclopentylmethyl-phenoxy)-1-((S)-...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Matrix metalloproteinase-3 by MCA peptide assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289672((R)-2-[(S)-3-(4-Isopropyl-phenoxy)-1-((S)-6-methyl...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Matrix metalloproteinase-3 by MCA peptide assayMore data for this Ligand-Target Pair
In DepthDetails Article