Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50030025
TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290345BDBM50290345(7-(3,4-Difluoro-benzyl)-1-(4-fluoro-phenyl)-4,5,6,...)
Affinity DataIC50: 2nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290353BDBM50290353([1-[1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,...)
Affinity DataIC50: 2.30nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290364BDBM50290364(7-Benzyl-1-(4-fluoro-phenyl)-4,5,6,7-tetrahydro-1H...)
Affinity DataIC50: 3nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290359BDBM50290359(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50: 3.20nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290336BDBM50290336(Acetic acid acetoxy-[1-(4-fluoro-phenyl)-7-naphtha...)
Affinity DataIC50: 5.30nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290361BDBM50290361(7-Naphthalen-1-ylmethyl-1-phenyl-4,5,6,7-tetrahydr...)
Affinity DataIC50: 6nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290333BDBM50290333(7-(4-Fluoro-benzyl)-1-(4-fluoro-phenyl)-4,5,6,7-te...)
Affinity DataIC50: 6.5nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290356BDBM50290356(1-(4-Fluoro-phenyl)-7-(4-methyl-benzyl)-4,5,6,7-te...)
Affinity DataIC50: 7.70nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290334BDBM50290334(1-(4-Chloro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50: 9nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290362BDBM50290362(7-(2-Chloro-benzyl)-1-(4-fluoro-phenyl)-4,5,6,7-te...)
Affinity DataIC50: 11nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290358BDBM50290358(7-(4-Chloro-benzyl)-1-(4-fluoro-phenyl)-4,5,6,7-te...)
Affinity DataIC50: 12nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290349BDBM50290349(1-(4-Methoxy-phenyl)-7-naphthalen-1-ylmethyl-4,5,6...)
Affinity DataIC50: 13nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290338BDBM50290338(1-(4-Fluoro-phenyl)-7-(3-methoxy-benzyl)-octahydro...)
Affinity DataIC50: 17nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290354BDBM50290354(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50: 41nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290375BDBM50290375(N-[1-[1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-...)
Affinity DataIC50: 49nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290360BDBM50290360([1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6...)
Affinity DataIC50: 52nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290372BDBM50290372(1-(4-Fluoro-phenyl)-7-naphthalen-2-ylmethyl-octahy...)
Affinity DataIC50: 56nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290368BDBM50290368(1-(3-Chloro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50: 69nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290352BDBM50290352(Acetic acid 1-(4-fluoro-phenyl)-7-naphthalen-1-ylm...)
Affinity DataIC50: 73nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290344BDBM50290344(Carbonic acid ethyl ester 1-(4-fluoro-phenyl)-7-na...)
Affinity DataIC50: 90nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290363BDBM50290363(3-[1,3]Dioxolan-2-yl-1-(4-fluoro-phenyl)-7-naphtha...)
Affinity DataIC50: 97nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290351BDBM50290351(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-3-viny...)
Affinity DataIC50: 147nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290376BDBM50290376(1-(4-Fluoro-phenyl)-7-(4-methoxy-benzyl)-4,5,6,7-t...)
Affinity DataIC50: 163nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290374BDBM50290374(Benzoic acid 1-(4-fluoro-phenyl)-7-naphthalen-1-yl...)
Affinity DataIC50: 182nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290369BDBM50290369(1-[1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5...)
Affinity DataIC50: 236nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290355BDBM50290355(N'-[1-[1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl...)
Affinity DataIC50: 547nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290343BDBM50290343(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50: 628nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290371BDBM50290371(1-[1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5...)
Affinity DataIC50: 690nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290337BDBM50290337(4-(3-Formyl-7-naphthalen-1-ylmethyl-4,5,6,7-tetrah...)
Affinity DataIC50: 851nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290335BDBM50290335(7-(4-tert-Butyl-benzyl)-1-(4-fluoro-phenyl)-4,5,6,...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290340BDBM50290340(1-[1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290350BDBM50290350(Diethyl-[1-(4-fluoro-phenyl)-7-naphthalen-1-ylmeth...)
Affinity DataIC50: 1.38E+3nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290370BDBM50290370(Benzyl-[1-(4-fluoro-phenyl)-7-naphthalen-1-ylmethy...)
Affinity DataIC50: 1.38E+3nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290347BDBM50290347([1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6...)
Affinity DataIC50: 1.57E+3nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290373BDBM50290373(1-[1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5...)
Affinity DataIC50: 1.76E+3nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290366BDBM50290366(7-(3,4-Dimethoxy-benzyl)-1-(4-fluoro-phenyl)-4,5,6...)
Affinity DataIC50: 1.89E+3nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290341BDBM50290341(1-(4-Fluoro-phenyl)-7-(4-isopropyl-benzyl)-4,5,6,7...)
Affinity DataIC50: 2.20E+3nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290342BDBM50290342(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290346BDBM50290346(Octanoic acid 1-(4-fluoro-phenyl)-7-naphthalen-1-y...)
Affinity DataIC50: 4.01E+3nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290367BDBM50290367(Acetic acid [1-[1-(4-fluoro-phenyl)-7-naphthalen-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290365BDBM50290365(1-(4-Fluoro-phenyl)-3-(N'-[(E)-methylene]benzenesu...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290339BDBM50290339(Benzoic acid [1-[1-(4-fluoro-phenyl)-7-naphthalen-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290357BDBM50290357(7-Biphenyl-4-ylmethyl-1-(4-fluoro-phenyl)-4,5,6,7-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290332BDBM50290332(4-(3-Formyl-7-naphthalen-1-ylmethyl-4,5,6,7-tetrah...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProgesterone receptor(Rabbit)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50290348BDBM50290348(1-(4-Fluoro-phenyl)-7-naphthalen-1-ylmethyl-4,5,6,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity determined by ability to displace [3H]R5020 radioligand using uterine progesterone receptor obtained from estrogen-primed rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article