Compile Data Set for Download or QSAR
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Found 13 Enz. Inhib. hit(s) with all data for entry = 50030054
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50089913(4-(Amino-carboxy-methyl)-2-hydroxy-3-methyl-benzoi...)
Affinity DataIC50:  6.00E+3nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR1-alpha expressed in AV-12 cells by measuring inhibitory co...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50084140(4-((S)-Amino-carboxy-methyl)-3-methyl-benzoic acid...)
Affinity DataIC50:  1.90E+4nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR1-alpha expressed in AV-12 cells by measuring inhibitory co...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50084140(4-((S)-Amino-carboxy-methyl)-3-methyl-benzoic acid...)
Affinity DataIC50:  1.90E+4nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR5a expressed in AV-12 cells by measuring inhibitory concent...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50053588((S)-4-(amino(carboxy)methyl)benzoic acid | (S)-4-c...)
Affinity DataIC50:  5.80E+4nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR1-alpha expressed in AV-12 cells by measuring inhibitory co...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290679(4-(Amino-carboxy-methyl)-2-hydroxy-5-methyl-benzoi...)
Affinity DataIC50:  7.30E+4nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR1-alpha expressed in AV-12 cells by measuring inhibitory co...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50089913(4-(Amino-carboxy-methyl)-2-hydroxy-3-methyl-benzoi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR5a expressed in AV-12 cells by measuring inhibitory concent...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50053588((S)-4-(amino(carboxy)methyl)benzoic acid | (S)-4-c...)
Affinity DataIC50:  1.55E+5nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR5a expressed in AV-12 cells by measuring inhibitory concent...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50030630((RS)-1-aminoindan-1,5-dicarboxylic acid | 1-Amino-...)
Affinity DataIC50:  2.14E+5nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR1-alpha expressed in AV-12 cells by measuring inhibitory co...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50084140(4-((S)-Amino-carboxy-methyl)-3-methyl-benzoic acid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR5a expressed in AV-12 cells by measuring inhibitory concent...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50084140(4-((S)-Amino-carboxy-methyl)-3-methyl-benzoic acid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR5a expressed in AV-12 cells by measuring inhibitory concent...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50084140(4-((S)-Amino-carboxy-methyl)-3-methyl-benzoic acid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR5a expressed in AV-12 cells by measuring inhibitory concent...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50084140(4-((S)-Amino-carboxy-methyl)-3-methyl-benzoic acid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR1-alpha expressed in AV-12 cells by measuring inhibitory co...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290679(4-(Amino-carboxy-methyl)-2-hydroxy-5-methyl-benzoi...)
Affinity DataIC50: >3.00E+5nMAssay Description:Compound was tested for functional response of human metabotropic glutamate receptor mGluR5a expressed in AV-12 cells by measuring inhibitory concent...More data for this Ligand-Target Pair
In DepthDetails Article