Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50030062
TargetTyrosine-protein kinase ZAP-70(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50069336(NQLPpYNELNLGRREEpYDVLD | NELNLGRREE | CHEMBL439120)
Affinity DataIC50: 30nMAssay Description:Antagonistic activity against SH2 domain of Zeta-chain (TCR) associated protein kinase, ZAP-70More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetTyrosine-protein kinase ZAP-70(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290773(Non-peptide bidentate ITAM analogue | CHEMBL443592)
Affinity DataIC50: 250nMAssay Description:Antagonistic activity against SH2 domain of Zeta-chain (TCR) associated protein kinase, ZAP-70More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetTyrosine-protein kinase ZAP-70(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290771(Non-peptide bidentate ITAM analogue | CHEMBL386787)
Affinity DataIC50: 320nMAssay Description:Antagonistic activity against SH2 domain of Zeta-chain (TCR) associated protein kinase, ZAP-70More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetTyrosine-protein kinase ZAP-70(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290774([Difluoro-(4-{[hexanoyl-((8R,9S,13S,14S,17S)-13-me...)
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonistic activity against SH2 domain of Zeta-chain (TCR) associated protein kinase, ZAP-70More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetTyrosine-protein kinase ZAP-70(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290772((4-{[Hexanoyl-((8R,9S,13S,14S,17S)-13-methyl-3-pro...)
Affinity DataIC50: 3.20E+3nMAssay Description:Antagonistic activity against SH2 domain of Zeta-chain (TCR) associated protein kinase, ZAP-70More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article