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Found 19 Enz. Inhib. hit(s) with all data for entry = 50031772
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318712((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  80nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318713((2S,15S,18S,21S,24S)-15-(3-amino-3-oxopropyl)-2-be...)
Affinity DataKi:  80nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318710((2S,15S,18S,21S,24S)-2,15-dibenzyl-24-carbamoyl-18...)
Affinity DataKi:  200nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318714((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  300nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318711((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  400nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318715((2S,15S,18S,21S,24S)-2-benzyl-24-carbamoyl-18,21-d...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318716((2S,8S,15S,18S,21S,24S)-2-benzyl-24-carbamoyl-18,2...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318712((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318717((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318709((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318714((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  1.24E+4nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318718((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  2.08E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318711((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  2.22E+4nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318710((2S,15S,18S,21S,24S)-2,15-dibenzyl-24-carbamoyl-18...)
Affinity DataKi:  2.29E+4nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318715((2S,15S,18S,21S,24S)-2-benzyl-24-carbamoyl-18,21-d...)
Affinity DataKi:  3.07E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318716((2S,8S,15S,18S,21S,24S)-2-benzyl-24-carbamoyl-18,2...)
Affinity DataKi:  3.36E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318710((2S,15S,18S,21S,24S)-2,15-dibenzyl-24-carbamoyl-18...)
Affinity DataKi:  3.48E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318712((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  3.75E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318717((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed