Compile Data Set for Download or QSAR
Report error Found 186 Enz. Inhib. hit(s) with all data for entry = 50031856
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320533BDBM50320533(3-(4-Methylbenzylidene)anabaseine | CHEMBL1163379)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320547BDBM50320547(3-(4-Difluoromethoxybenzylidene)anabaseine | CHEMB...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320533BDBM50320533(3-(4-Methylbenzylidene)anabaseine | CHEMBL1163379)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320547BDBM50320547(3-(4-Difluoromethoxybenzylidene)anabaseine | CHEMB...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320544BDBM50320544(3-(3-(4-chlorobenzylidene)-3,4,5,6-tetrahydropyrid...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320544BDBM50320544(3-(3-(4-chlorobenzylidene)-3,4,5,6-tetrahydropyrid...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320551BDBM50320551(3-(4-Trifluoromethoxybenzylidene)anabaseine | CHEM...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320551BDBM50320551(3-(4-Trifluoromethoxybenzylidene)anabaseine | CHEM...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320551BDBM50320551(3-(4-Trifluoromethoxybenzylidene)anabaseine | CHEM...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320551BDBM50320551(3-(4-Trifluoromethoxybenzylidene)anabaseine | CHEM...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320535BDBM50320535(3-(4-Acetylbenzylidene)anabaseine | CHEMBL1164787)
Affinity DataKi:  36nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320535BDBM50320535(3-(4-Acetylbenzylidene)anabaseine | CHEMBL1164787)
Affinity DataKi:  36nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320539BDBM50320539(3-(4-n-Butoxybenzylidene)anabaseine | CHEMBL116546...)
Affinity DataKi:  41nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320539BDBM50320539(3-(4-n-Butoxybenzylidene)anabaseine | CHEMBL116546...)
Affinity DataKi:  41nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320525BDBM50320525(3-(4-Methylthiobenzylidene)anabaseine | CHEMBL1165...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320525BDBM50320525(3-(4-Methylthiobenzylidene)anabaseine | CHEMBL1165...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320552BDBM50320552(3-(4-n-Propylbenzylidene)anabaseine | CHEMBL116468...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320552BDBM50320552(3-(4-n-Propylbenzylidene)anabaseine | CHEMBL116468...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320563BDBM50320563(3-(2,4,6-Trimethoxybenzylidene)anabaseine | CHEMBL...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320563BDBM50320563(3-(2,4,6-Trimethoxybenzylidene)anabaseine | CHEMBL...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264117BDBM50264117(3-[1-(4-Hydroxy-2-methoxy-phenyl)-meth-(E)-ylidene...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50264117BDBM50264117(3-[1-(4-Hydroxy-2-methoxy-phenyl)-meth-(E)-ylidene...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320546BDBM50320546(3-(4-Pivaloyloxybenzylidene)anabaseine | CHEMBL116...)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320546BDBM50320546(3-(4-Pivaloyloxybenzylidene)anabaseine | CHEMBL116...)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320528BDBM50320528(3-(2-Hydroxy-4-diethylaminobenzylidene)anabaseine ...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320528BDBM50320528(3-(2-Hydroxy-4-diethylaminobenzylidene)anabaseine ...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320545BDBM50320545(3-(2-acetoxylbenzylidine)anabasaine | CHEMBL116521...)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320545BDBM50320545(3-(2-acetoxylbenzylidine)anabasaine | CHEMBL116521...)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320546BDBM50320546(3-(4-Pivaloyloxybenzylidene)anabaseine | CHEMBL116...)
Affinity DataKi:  161nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320546BDBM50320546(3-(4-Pivaloyloxybenzylidene)anabaseine | CHEMBL116...)
Affinity DataKi:  161nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320555BDBM50320555(3-(2-Pivaloyloxybenzylidene)anabaseine | CHEMBL116...)
Affinity DataKi:  187nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320555BDBM50320555(3-(2-Pivaloyloxybenzylidene)anabaseine | CHEMBL116...)
Affinity DataKi:  187nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320567BDBM50320567(3-(2,4-Dihydroxybenzylidene)anabaseine | CHEMBL116...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320567BDBM50320567(3-(2,4-Dihydroxybenzylidene)anabaseine | CHEMBL116...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320548BDBM50320548(3-(3-benzylidene-3,4,5,6-tetrahydropyridin-2-yl)py...)
Affinity DataKi:  222nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320548BDBM50320548(3-(3-benzylidene-3,4,5,6-tetrahydropyridin-2-yl)py...)
Affinity DataKi:  222nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320545BDBM50320545(3-(2-acetoxylbenzylidine)anabasaine | CHEMBL116521...)
Affinity DataKi:  244nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320545BDBM50320545(3-(2-acetoxylbenzylidine)anabasaine | CHEMBL116521...)
Affinity DataKi:  244nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320564BDBM50320564(3-(4-Methoxybenzylidene)anabaseine | CHEMBL1164117)
Affinity DataKi:  244nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320564BDBM50320564(3-(4-Methoxybenzylidene)anabaseine | CHEMBL1164117)
Affinity DataKi:  244nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061564BDBM50061564(3-[1-(2,4-Dimethoxy-phenyl)-meth-(E)-ylidene]-3,4,...)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50061564BDBM50061564(3-[1-(2,4-Dimethoxy-phenyl)-meth-(E)-ylidene]-3,4,...)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320554BDBM50320554(3-(3,5-Dimethyl-4-hydroxybenzylidene)anabaseine | ...)
Affinity DataKi:  276nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320554BDBM50320554(3-(3,5-Dimethyl-4-hydroxybenzylidene)anabaseine | ...)
Affinity DataKi:  276nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320550BDBM50320550(3-[4-(1H-1,2,4-Triazol-1-yl)benzylidene]anabaseine...)
Affinity DataKi:  284nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320550BDBM50320550(3-[4-(1H-1,2,4-Triazol-1-yl)benzylidene]anabaseine...)
Affinity DataKi:  284nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320564BDBM50320564(3-(4-Methoxybenzylidene)anabaseine | CHEMBL1164117)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320564BDBM50320564(3-(4-Methoxybenzylidene)anabaseine | CHEMBL1164117)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320553BDBM50320553(3-(3-Methoxybenzylidene)anabaseine | CHEMBL1164724)
Affinity DataKi:  337nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Florida

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50320553BDBM50320553(3-(3-Methoxybenzylidene)anabaseine | CHEMBL1164724)
Affinity DataKi:  337nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
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