Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50033070
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339101BDBM50339101(5-(aminomethyl)-4-(2,4-dichlorophenyl)-N,6-dimethy...)
Affinity DataIC50: 6nMAssay Description:Competitive inhibition of human recombinant DPP4 by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339103BDBM50339103(5-Aminomethyl-4-(2,4-dichlorophenyl)-6-methyl-pyri...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339101BDBM50339101(5-(aminomethyl)-4-(2,4-dichlorophenyl)-N,6-dimethy...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339100BDBM50339100(5-(aminomethyl)-4-(2,4-dichlorophenyl)-6-methylpic...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339102BDBM50339102((5-(aminomethyl)-4-(2,4-dichlorophenyl)-6-methylpy...)
Affinity DataIC50: 44nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339095BDBM50339095(5-(aminomethyl)-N-cyclopropyl-4-(4-fluorophenyl)-6...)
Affinity DataIC50: 80nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339098BDBM50339098(5-(aminomethyl)-N-cyclopropyl-4-(2,4-difluoropheny...)
Affinity DataIC50: 674nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339099BDBM50339099(5-(aminomethyl)-4-(2,4-difluorophenyl)-6-methyl-N-...)
Affinity DataIC50: 674nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339096BDBM50339096((5-(aminomethyl)-4-(4-fluorophenyl)-6-methylpyridi...)
Affinity DataIC50: 686nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339097BDBM50339097(ethyl 1-(5-(aminomethyl)-4-(4-fluorophenyl)-6-meth...)
Affinity DataIC50: 937nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229666BDBM50229666(Ile-Pro-Ile | (2S,3S)-2-((S)-1-((2S,3S)-2-amino-3-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339102BDBM50339102((5-(aminomethyl)-4-(2,4-dichlorophenyl)-6-methylpy...)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339100BDBM50339100(5-(aminomethyl)-4-(2,4-dichlorophenyl)-6-methylpic...)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339101BDBM50339101(5-(aminomethyl)-4-(2,4-dichlorophenyl)-N,6-dimethy...)
Affinity DataKi:  3.90E+4nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50229666BDBM50229666(Ile-Pro-Ile | (2S,3S)-2-((S)-1-((2S,3S)-2-amino-3-...)
Affinity DataKi:  3.90E+4nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339108BDBM50339108(5-(aminomethyl)-4-(4-methoxyphenyl)-6-methyl-N-(5-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339109BDBM50339109((R)-(5-(aminomethyl)-4-(4-methoxyphenyl)-6-methylp...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339110BDBM50339110((5-(aminomethyl)-4-(4-methoxyphenyl)-6-methylpyrid...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339111BDBM50339111(5-(aminomethyl)-4-(4-methoxyphenyl)-6-methyl-N-(2-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339104BDBM50339104(5-(aminomethyl)-N-cyclopropyl-4-(4-methoxyphenyl)-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339105BDBM50339105((5-(aminomethyl)-4-(4-methoxyphenyl)-6-methylpyrid...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339106BDBM50339106((5-(aminomethyl)-4-(4-methoxyphenyl)-6-methylpyrid...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339107BDBM50339107(5-(aminomethyl)-N-(3,4-dichlorobenzyl)-4-(4-methox...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339116BDBM50339116((3-(aminomethyl)-6-(4-fluorophenyl)-2-methylpyridi...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339117BDBM50339117((3-(aminomethyl)-6-(4-chlorophenyl)-2-methylpyridi...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339118BDBM50339118((3-(aminomethyl)-6-(4-chlorophenyl)-2-methylpyridi...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339119BDBM50339119(ethyl 1-(3-(aminomethyl)-6-(4-chlorophenyl)-2-meth...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339112BDBM50339112(6-(aminomethyl)-4-(2-fluorophenyl)-2-methylnicotin...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339113BDBM50339113(6-(aminomethyl)-4-(4-chlorophenyl)-2-methylnicotin...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339114BDBM50339114(6-(aminomethyl)-4-(2,4-dichlorophenyl)-2-methylnic...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339115BDBM50339115(6-(aminomethyl)-4-(4-methoxyphenyl)-2-methylnicoti...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339124BDBM50339124((3-(aminomethyl)-6-(4-methoxyphenyl)-2-methylpyrid...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339125BDBM50339125((3-(aminomethyl)-6-(4-methoxyphenyl)-2-methylpyrid...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339093BDBM50339093(5-cyano-4-(2,4-dichlorophenyl)-6-methylpicolinamid...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339094BDBM50339094(5-cyano-4-(2,4-dichlorophenyl)-N,6-dimethylpicolin...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339120BDBM50339120(3-(aminomethyl)-N-cyclopropyl-6-(2,4-dichloropheny...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339121BDBM50339121((3-(aminomethyl)-6-(2,4-dichlorophenyl)-2-methylpy...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339122BDBM50339122((3-(aminomethyl)-6-(2,4-dichlorophenyl)-2-methylpy...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339123BDBM50339123(3-(aminomethyl)-N-cyclopropyl-6-(4-methoxyphenyl)-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DPP4 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339103BDBM50339103(5-Aminomethyl-4-(2,4-dichlorophenyl)-6-methyl-pyri...)
Affinity DataKi:  6.60E+4nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339095BDBM50339095(5-(aminomethyl)-N-cyclopropyl-4-(4-fluorophenyl)-6...)
Affinity DataKi:  1.06E+5nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339096BDBM50339096((5-(aminomethyl)-4-(4-fluorophenyl)-6-methylpyridi...)
Affinity DataKi:  1.37E+5nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339099BDBM50339099(5-(aminomethyl)-4-(2,4-difluorophenyl)-6-methyl-N-...)
Affinity DataKi:  1.79E+5nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50339098BDBM50339098(5-(aminomethyl)-N-cyclopropyl-4-(2,4-difluoropheny...)
Affinity DataKi:  1.82E+5nMAssay Description:Inhibition of human recombinant DPP8 assessed as Gly-Pro-pNA chromogenic substrate cleavage for 16 mins preincubated with compound for 10 mins before...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed