Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50033649
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20732BDBM20732(geldanomycin | GM-BODIPY | Geldanamycin | CHEMBL27...)
Affinity DataIC50: 40nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349038BDBM50349038(CHEMBL1807797)
Affinity DataIC50: 58nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349047BDBM50349047(CHEMBL1807807)
Affinity DataIC50: 60nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349032BDBM50349032(CHEMBL1807791)
Affinity DataIC50: 64nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349045BDBM50349045(CHEMBL1807805)
Affinity DataIC50: 65nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349042BDBM50349042(CHEMBL1807801)
Affinity DataIC50: 66nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349050BDBM50349050(CHEMBL1807810)
Affinity DataIC50: 68nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349046BDBM50349046(CHEMBL1807806)
Affinity DataIC50: 70nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349040BDBM50349040(CHEMBL1807799)
Affinity DataIC50: 74nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349041BDBM50349041(CHEMBL1807800)
Affinity DataIC50: 77nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349052BDBM50349052(CHEMBL1806511)
Affinity DataIC50: 80nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349039BDBM50349039(CHEMBL1807798)
Affinity DataIC50: 81nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349031BDBM50349031(CHEMBL1807790)
Affinity DataIC50: 82nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349049BDBM50349049(CHEMBL1807809)
Affinity DataIC50: 83nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349030BDBM50349030(CHEMBL1807804)
Affinity DataIC50: 83nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349044BDBM50349044(CHEMBL1807803)
Affinity DataIC50: 83nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349036BDBM50349036(CHEMBL1807795)
Affinity DataIC50: 84nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349037BDBM50349037(CHEMBL1807796)
Affinity DataIC50: 85nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349034BDBM50349034(CHEMBL1807793)
Affinity DataIC50: 88nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349054BDBM50349054(CHEMBL1807813)
Affinity DataIC50: 91nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50345151BDBM50345151(CHEMBL1779531)
Affinity DataIC50: 96nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340250BDBM50340250((6S)-6,15,15,18-tetramethyl-17-oxo-2,3,4,5,6,7,14,...)
Affinity DataIC50: 110nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349048BDBM50349048(CHEMBL1807808)
Affinity DataIC50: 116nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349033BDBM50349033(CHEMBL1807792)
Affinity DataIC50: 116nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349043BDBM50349043(CHEMBL1807802)
Affinity DataIC50: 131nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349035BDBM50349035(CHEMBL1807794)
Affinity DataIC50: 142nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349055BDBM50349055(CHEMBL1778194)
Affinity DataIC50: 145nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349053BDBM50349053(CHEMBL1807812)
Affinity DataIC50: 183nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50340251BDBM50340251(CHEMBL1760603)
Affinity DataIC50: 210nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50349051BDBM50349051(CHEMBL1807811)
Affinity DataIC50: 228nMAssay Description:Binding affinity to HSP90alpha after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50349030BDBM50349030(CHEMBL1807804)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed