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Found 47 Enz. Inhib. hit(s) with all data for entry = 50034473
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363052(CHEMBL1946956)
Affinity DataIC50:  400nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363017(CHEMBL1945812)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50343350(4,4,4-trifluoro-1-(4-(3-(thiophen-2-yl)-1,2,4-oxad...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50343351(4,4,4-Trifluoro-1-[(R)-3-(3-thiophen-2-yl-1,2,4-ox...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363015(CHEMBL1945701)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363018(CHEMBL1945813)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363019(CHEMBL1945814)
Affinity DataEC50:  2.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363020(CHEMBL1945815)
Affinity DataEC50:  9.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363021(CHEMBL1945816)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363022(CHEMBL1945817)
Affinity DataEC50:  4.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363023(CHEMBL1945818)
Affinity DataEC50:  9.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363024(CHEMBL1945819)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363025(CHEMBL1945820)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363026(CHEMBL1944650)
Affinity DataEC50:  7.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363027(CHEMBL1945821)
Affinity DataEC50:  6.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363028(CHEMBL1945961)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363029(CHEMBL1945962)
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363030(CHEMBL1945963)
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363031(CHEMBL1945964)
Affinity DataEC50:  2.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363032(CHEMBL1945965)
Affinity DataEC50:  2.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363033(CHEMBL1945966)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363034(CHEMBL1945967)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363035(CHEMBL1945968)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363036(CHEMBL1945969)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363037(CHEMBL1945970)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363038(CHEMBL1945971)
Affinity DataEC50:  2.50E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363039(CHEMBL1945972)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363040(CHEMBL1946415)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363041(CHEMBL1946416)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363042(CHEMBL1946417)
Affinity DataEC50:  800nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363043(CHEMBL1946418)
Affinity DataEC50:  4.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363044(CHEMBL1946419)
Affinity DataEC50:  800nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363045(CHEMBL1946420)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363046(CHEMBL1946421)
Affinity DataEC50: >5.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363047(CHEMBL1946422)
Affinity DataEC50:  3.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363048(CHEMBL1946423)
Affinity DataEC50: >5.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363049(CHEMBL1946424)
Affinity DataEC50:  4.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363050(CHEMBL1946425)
Affinity DataEC50: >5.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363051(CHEMBL1946426)
Affinity DataEC50:  6.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363052(CHEMBL1946956)
Affinity DataEC50:  60nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363018(CHEMBL1945813)
Affinity DataEC50:  500nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363017(CHEMBL1945812)
Affinity DataEC50:  200nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363016(CHEMBL1945811)
Affinity DataEC50:  2.50E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363015(CHEMBL1945701)
Affinity DataEC50:  500nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363014(CHEMBL1945700)
Affinity DataEC50:  1.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50343351(4,4,4-Trifluoro-1-[(R)-3-(3-thiophen-2-yl-1,2,4-ox...)
Affinity DataEC50:  400nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis)
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50343350(4,4,4-trifluoro-1-(4-(3-(thiophen-2-yl)-1,2,4-oxad...)
Affinity DataEC50:  100nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed