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Found 16 Enz. Inhib. hit(s) with all data for entry = 50034723
TargetKappa-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280516(2-(3,4-Dichloro-phenyl)-N-((1S,2S)-5-methoxy-2-pyr...)
Affinity DataKi:  6nMAssay Description:Compound was evaluated for the binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280515(2-(3,4-Dichloro-phenyl)-N-methyl-N-((1S,2S)-2-pyrr...)
Affinity DataKi:  10nMAssay Description:Compound was evaluated for the binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  15nMAssay Description:Compound was evaluated for the binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  38nMAssay Description:Compound was evaluated for the binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  51nMAssay Description:Compound was evaluated for the binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280516(2-(3,4-Dichloro-phenyl)-N-((1S,2S)-5-methoxy-2-pyr...)
Affinity DataKi:  304nMAssay Description:Compound was evaluated for the binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280515(2-(3,4-Dichloro-phenyl)-N-methyl-N-((1S,2S)-2-pyrr...)
Affinity DataKi:  545nMAssay Description:Compound was evaluated for the binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  696nMAssay Description:Compound was evaluated for the binding affinity to sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  825nMAssay Description:Compound was evaluated for the binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  1.90E+3nMAssay Description:Compound was evaluated for the binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280516(2-(3,4-Dichloro-phenyl)-N-((1S,2S)-5-methoxy-2-pyr...)
Affinity DataKi:  2.09E+3nMAssay Description:Compound was evaluated for the binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280516(2-(3,4-Dichloro-phenyl)-N-((1S,2S)-5-methoxy-2-pyr...)
Affinity DataKi:  5.16E+3nMAssay Description:Compound was evaluated for the binding affinity to sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280515(2-(3,4-Dichloro-phenyl)-N-methyl-N-((1S,2S)-2-pyrr...)
Affinity DataKi:  1.00E+4nMAssay Description:Compound was evaluated for the binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for the binding affinity to sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280515(2-(3,4-Dichloro-phenyl)-N-methyl-N-((1S,2S)-2-pyrr...)
Affinity DataKi:  1.00E+4nMAssay Description:Compound was evaluated for the binding affinity to sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  2.10E+4nMAssay Description:Compound was evaluated for the binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article