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Found 66 Enz. Inhib. hit(s) with all data for entry = 50034889
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289794(CHEMBL292119 | [2-(1H-Indol-3-yl)-1-isobutylcarbam...)
Affinity DataKi:  37nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289823(CHEMBL418299 | {(S)-2-(1H-Indol-3-yl)-1-[2-(1H-ind...)
Affinity DataKi:  980nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289798(CHEMBL59187 | [(S)-2-(1H-Indol-3-yl)-1-phenethylca...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289801(CHEMBL292766 | [(S)-2-(1H-Indol-3-yl)-1-phenethylc...)
Affinity DataKi:  2.60E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289822(CHEMBL291924 | [2-(1H-Indol-3-yl)-1-phenethylcarba...)
Affinity DataKi:  2.60E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289834(CHEMBL60125 | [(S)-2-(1H-Indol-3-yl)-1-(3-methyl-b...)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289829(CHEMBL291925 | [(S)-2-(1H-Indol-3-yl)-1-phenethylc...)
Affinity DataKi:  2.70E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289827(CHEMBL59561 | {(S)-2-(1H-Indol-3-yl)-1-[2-(1H-indo...)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289850(CHEMBL59055 | [(S)-2-(1H-Indol-3-yl)-1-isobutylcar...)
Affinity DataKi:  3.50E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289833(CHEMBL294165 | {(S)-2-(1H-Indol-3-yl)-1-[2-(1H-ind...)
Affinity DataKi:  3.70E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289799(CHEMBL293240 | [(S)-2-(1H-Indol-3-yl)-1-(3-methyl-...)
Affinity DataKi:  3.90E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289799(CHEMBL293240 | [(S)-2-(1H-Indol-3-yl)-1-(3-methyl-...)
Affinity DataKi:  3.90E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289808(CHEMBL61615 | [(S)-2-(1H-Indol-3-yl)-1-phenethylca...)
Affinity DataKi:  4.30E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289825(CHEMBL59060 | {(S)-2-(1H-Indol-3-yl)-1-[2-(1H-indo...)
Affinity DataKi:  4.70E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289837(CHEMBL61098 | [1-[2-(1H-Imidazol-4-yl)-ethylcarbam...)
Affinity DataKi:  5.00E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289809(CHEMBL58852 | [(S)-2-(1H-Indol-3-yl)-1-(3-methyl-b...)
Affinity DataKi:  6.10E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289814(CHEMBL60176 | [(S)-1-(5-Amino-pentylcarbamoyl)-2-(...)
Affinity DataKi:  7.80E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289810(CHEMBL301636 | {(S)-2-(1H-Indol-3-yl)-1-[2-(1H-ind...)
Affinity DataKi:  8.90E+3nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289793(CHEMBL61351 | [1-[2-(1H-Imidazol-4-yl)-ethylcarbam...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289795(CHEMBL61237 | [(S)-2-(1H-Indol-3-yl)-1-isobutylcar...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289796(3-{(S)-3-(1H-Indol-3-yl)-2-[2-(1H-indol-3-yl)-etho...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289797(CHEMBL59178 | [(S)-1-(5-Amino-pentylcarbamoyl)-2-(...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289802(CHEMBL57951 | [(S)-1-(2-Hydroxy-ethylcarbamoyl)-2-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289800(CHEMBL61041 | [(S)-2-(1H-Indol-3-yl)-1-phenethylca...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289803(CHEMBL59382 | [(S)-2-(1H-Indol-3-yl)-1-isobutylcar...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289805(CHEMBL432510 | {(S)-2-(1H-Indol-3-yl)-1-[2-(1H-ind...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289804(CHEMBL300578 | [(S)-2-(1H-Indol-3-yl)-1-phenethylc...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289806(CHEMBL59243 | [1-[2-(1H-Imidazol-4-yl)-ethylcarbam...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289811(CHEMBL58442 | [1-[2-(1H-Imidazol-4-yl)-ethylcarbam...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289812(CHEMBL61183 | [(S)-2-(1H-Indol-3-yl)-1-isobutylcar...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289813(CHEMBL59246 | [1-[2-(1H-Imidazol-4-yl)-ethylcarbam...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289815(CHEMBL59519 | [(S)-1-(5-Amino-pentylcarbamoyl)-2-(...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289818(CHEMBL58605 | [(S)-2-(1H-Indol-3-yl)-1-(3-methyl-b...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289817(3-[(S)-3-(1H-Indol-3-yl)-2-methoxycarbonylamino-pr...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289816(CHEMBL300380 | [(S)-1-(2-Hydroxy-ethylcarbamoyl)-2...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289820(CHEMBL58537 | [(S)-1-(5-Amino-pentylcarbamoyl)-2-(...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289819(CHEMBL301849 | [1-[2-(1H-Imidazol-4-yl)-ethylcarba...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289821(CHEMBL58851 | [(S)-1-(5-Amino-pentylcarbamoyl)-2-(...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289831(CHEMBL293281 | [(S)-2-(1H-Indol-3-yl)-1-isobutylca...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289824(CHEMBL304238 | [(S)-1-(2-Hydroxy-ethylcarbamoyl)-2...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289828(CHEMBL58400 | [(S)-2-(1H-Indol-3-yl)-1-(3-methyl-b...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289826(CHEMBL299689 | {(S)-2-(1H-Indol-3-yl)-1-[2-(1H-ind...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289830(CHEMBL58868 | [(S)-1-(2-Hydroxy-ethylcarbamoyl)-2-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289832(CHEMBL300374 | [(S)-1-(5-Amino-pentylcarbamoyl)-2-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289839(CHEMBL59513 | [(S)-2-(1H-Indol-3-yl)-1-isobutylcar...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289836(CHEMBL58167 | [(S)-2-(1H-Indol-3-yl)-1-phenethylca...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289835(CHEMBL431327 | [(S)-1-(5-Amino-pentylcarbamoyl)-2-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289840(CHEMBL59777 | [(S)-2-(1H-Indol-3-yl)-1-phenethylca...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289841(CHEMBL57599 | [(S)-2-(1H-Indol-3-yl)-1-isobutylcar...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289838(3-[(S)-2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human neuromedin B(hNMB) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
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