Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50034994
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50087097BDBM50087097(1-{[2-(1-Carboxy-2-phenyl-ethylcarbamoyl)-3-phenyl...)
Affinity DataKi:  2.20nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for A+B stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078127BDBM50078127(2-{3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoy...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078134BDBM50078134(2-{3-[(1-Amino-2-phenyl-ethyl)-hydroxy-phosphinoyl...)
Affinity DataKi:  2.90nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for A+B stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078131BDBM50078131(2-{3-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyl...)
Affinity DataKi:  3.20nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for A+B stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078135BDBM50078135(2-{3-[(Amino-phenyl-methyl)-hydroxy-phosphinoyl]-2...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078137BDBM50078137(2-{3-[(1-Amino-3-methylsulfanyl-propyl)-hydroxy-ph...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078128BDBM50078128((S)-2-Amino-4-methylsulfanyl-butane-1-thiol | CHEM...)
Affinity DataKi:  11nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078133BDBM50078133(2-Amino-4-methyl-pentane-1-thiol | (S)-2-Amino-4-m...)
Affinity DataKi:  22nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078138BDBM50078138((S)-2-Amino-2-phenyl-ethanethiol | CHEMBL286865)
Affinity DataKi:  25nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078121BDBM50078121((S)-2-Amino-4-phenyl-butane-1-thiol | CHEMBL34963)
Affinity DataKi:  27nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078126BDBM50078126((S)-2-Amino-propane-1-thiol | CHEMBL37279)
Affinity DataKi:  28nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078129BDBM50078129((S)-2-Amino-3-phenyl-propane-1-thiol | 2-Amino-3-p...)
Affinity DataKi:  30nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078131BDBM50078131(2-{3-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyl...)
Affinity DataKi:  90nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for C+D stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078125BDBM50078125((1-Amino-3-phenyl-propyl)-phosphinic acid | CHEMBL...)
Affinity DataKi:  130nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21460BDBM21460(CHEMBL34068 | 3-[(1-amino-2-phenylethyl)(hydroxy)p...)
Affinity DataKi:  190nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078134BDBM50078134(2-{3-[(1-Amino-2-phenyl-ethyl)-hydroxy-phosphinoyl...)
Affinity DataKi:  200nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for C+D stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078135BDBM50078135(2-{3-[(Amino-phenyl-methyl)-hydroxy-phosphinoyl]-2...)
Affinity DataKi:  320nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for C+D stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078127BDBM50078127(2-{3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoy...)
Affinity DataKi:  360nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for C+D stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21461BDBM21461(CHEMBL36716 | 3-[(1-amino-3-methylbutyl)(hydroxy)p...)
Affinity DataKi:  370nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078137BDBM50078137(2-{3-[(1-Amino-3-methylsulfanyl-propyl)-hydroxy-ph...)
Affinity DataKi:  370nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for C+D stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078130BDBM50078130((1-Amino-3-methylsulfanyl-propyl)-phosphinic acid ...)
Affinity DataKi:  400nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50087097BDBM50087097(1-{[2-(1-Carboxy-2-phenyl-ethylcarbamoyl)-3-phenyl...)
Affinity DataKi:  670nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for C+D stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078139BDBM50078139((1-Ammonium-2-phenyl-ethyl)-phosphinic acid | (1-A...)
Affinity DataKi:  960nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078132BDBM50078132((1-Amino-3-methyl-butyl)-phosphinic acid | (1-Ammo...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078136BDBM50078136((Amino-phenyl-methyl)-phosphinic acid | CHEMBL3997...)
Affinity DataKi:  4.80E+3nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078124BDBM50078124((1-Amino-ethyl)-phosphinic acid | CHEMBL37702)
Affinity DataKi:  8.40E+3nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078122BDBM50078122((R)-1-{[(S)-2-((S)-1-Carboxy-1-methyl-2-phenyl-eth...)
Affinity DataKi:  0nMAssay Description:Inhibitory activity was measured on Aminopeptidase using GluNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078122BDBM50078122((R)-1-{[(S)-2-((S)-1-Carboxy-1-methyl-2-phenyl-eth...)
Affinity DataKi:  0nMAssay Description:Inhibitory activity was measured on Aminopeptidase N using Ala-p.NA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078120BDBM50078120((R)-1-{[(S)-2-((S)-1-Carboxy-1-methyl-2-phenyl-eth...)
Affinity DataKi:  0nMAssay Description:Inhibitory activity was measured on Aminopeptidase N using Ala-p.NA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Mouse)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078120BDBM50078120((R)-1-{[(S)-2-((S)-1-Carboxy-1-methyl-2-phenyl-eth...)
Affinity DataKi: >0nMAssay Description:Inhibitory activity was measured on Aminopeptidase B using Arg p.NA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamyl aminopeptidase(Pig)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078120BDBM50078120((R)-1-{[(S)-2-((S)-1-Carboxy-1-methyl-2-phenyl-eth...)
Affinity DataKi:  0nMAssay Description:Inhibitory activity was measured on Aminopeptidase using GluNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Mouse)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50078122BDBM50078122((R)-1-{[(S)-2-((S)-1-Carboxy-1-methyl-2-phenyl-eth...)
Affinity DataKi: >0nMAssay Description:Inhibitory activity was measured on Aminopeptidase B using Arg p.NA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed