Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50036059
TargetGamma-aminobutyric acid receptor subunit alpha-1(Mouse)
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001561BDBM50001561(CHEMBL132060 | 5-(6-Imino-3-thiophen-3-yl-6H-pyrid...)
Affinity DataIC50: 88nMAssay Description:Affinity for gamma-aminobutyric-acid A receptor measured by its ability to displace [3H]gabazine antagonist from rat brain preparations.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Mouse)
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001562BDBM50001562(CHEMBL552953 | 5-(6-Imino-3-phenyl-6H-pyridazin-1-...)
Affinity DataIC50: 240nMAssay Description:Affinity for gamma-aminobutyric-acid A receptor measured by its ability to displace [3H]gabazine antagonist from rat brain preparations.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Mouse)
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001556BDBM50001556(CHEMBL132561 | 4-(6-Imino-5-methyl-3-phenyl-6H-pyr...)
Affinity DataIC50: 800nMAssay Description:Affinity for gamma-aminobutyric-acid A receptor measured by its ability to displace [3H]gabazine antagonist from rat brain preparations.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed