Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50037717
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184615BDBM50184615((4aS,6aS,6bR,10S,12aR,14bS,E)-10-(3-(4-chloropheny...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184619BDBM50184619((4aS,6aS,6bR,12aR,14bS,E)-benzyl 11-(hydroxymethyl...)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184613BDBM50184613((4aS,6aS,6bR,12aR,14bS,E)-benzyl 11-(2,4-dichlorob...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184601BDBM50184601((4aS,6aS,6bR,13aR,15bS)-2,2,6a,6b,9,9,13a-heptamet...)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184618BDBM50184618((4aS,6aS,6bR,13aR,15bS)-2,2,6a,6b,9,9,13a-heptamet...)
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50346601BDBM50346601(Oleanolic acid (OA)(Compound 1) | NSC-114945 | OLE...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184603BDBM50184603((4aS,6aS,6bR,10S,12aR,14bS,E)-10-(3-(4-methoxyphen...)
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50346613BDBM50346613(Oleanonic Acid | CHEMBL470029)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184600BDBM50184600((4aS,6aS,6bR,13aR,15bS)-benzyl 2,2,6a,6b,9,9,13a-h...)
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184605BDBM50184605((4aS,6aS,6bR,12aR,14bS,E)-benzyl 10-(hydroxyimino)...)
Affinity DataIC50: 2.08E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184604BDBM50184604((4aS,6aS,6bR,10Z,11E,12aR,14bS)-benzyl 10,11-bis(h...)
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184614BDBM50184614((4aS,6aS,6bR,12aR,14bS,E)-11-(hydroxyimino)-2,2,6a...)
Affinity DataIC50: 2.61E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184611BDBM50184611((4aS,6aS,6bR,10R,12aR,14bS,E)-10-hydroxy-11-(hydro...)
Affinity DataIC50: 2.82E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184602BDBM50184602((4aS,6aS,6bR,10S,12aR,14bS)-10-(3-carboxypropanoyl...)
Affinity DataIC50: 3.43E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184598BDBM50184598((4aS,6aS,6bR,12aR,14bS,E)-benzyl 11-(hydroxyimino)...)
Affinity DataIC50: 4.68E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184607BDBM50184607((4aS,6aS,6bR,10S,12aR,14bS)-2-(methylamino)ethyl 1...)
Affinity DataIC50: 5.32E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184610BDBM50184610((4aS,6aS,6bR,12aR,14bS,E)-benzyl 11-(benzyloxyimin...)
Affinity DataIC50: 6.13E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184608BDBM50184608(2-((4aS,6aS,6bR,10S,12aR,14bS)-10-hydroxy-2,2,6a,6...)
Affinity DataIC50: 6.26E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184599BDBM50184599((4aS,6aS,6bR,12aR,14bS)-benzyl 2,2,6a,6b,9,9,12a-h...)
Affinity DataIC50: 6.66E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184609BDBM50184609((4aS,6aS,6bR,10S,12aR,14bS)-4-ethoxy-4-oxobutyl 10...)
Affinity DataIC50: 7.67E+4nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 10849BDBM10849(CHEMBL113 | 1,3,7-trimethyl-3,7-dihydropurine-2,6-...)
Affinity DataIC50: 1.14E+5nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184606BDBM50184606((4aS,6aS,6bR,10R,12aR,14bS,E)-benzyl 10-hydroxy-11...)
Affinity DataIC50: 1.79E+5nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184616BDBM50184616((4aS,6aS,6bR,12aR,14bS,E)-10-(hydroxyimino)-2,2,6a...)
Affinity DataIC50: 2.25E+5nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184617BDBM50184617((4aS,6aS,6bR,10S,12aR,14bS)-benzyl 10-hydroxy-2,2,...)
Affinity DataIC50: 4.61E+5nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50184612BDBM50184612(benzyl 2,2,6a,6b,9,9,13a-heptamethyl-1,2,3,4,4a,5,...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed