Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50038303
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374555BDBM50374555(REGRELOR DISODIUM)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374558BDBM50374558(CHEMBL255350)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374572BDBM50374572(CHEMBL403010)
Affinity DataIC50: 201nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374559BDBM50374559(CHEMBL255349)
Affinity DataIC50: 243nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374571BDBM50374571(CHEMBL272113)
Affinity DataIC50: 495nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374566BDBM50374566(CHEMBL272975)
Affinity DataIC50: 513nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374568BDBM50374568(CHEMBL401780)
Affinity DataIC50: 580nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374557BDBM50374557(CHEMBL267283)
Affinity DataIC50: 616nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374560BDBM50374560(CHEMBL256251)
Affinity DataIC50: 663nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374574BDBM50374574(CHEMBL265707)
Affinity DataIC50: 1.27E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374556BDBM50374556(CHEMBL412171)
Affinity DataIC50: 1.31E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374565BDBM50374565(CHEMBL403011)
Affinity DataIC50: 2.23E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374561BDBM50374561(CHEMBL427723)
Affinity DataIC50: 2.48E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374564BDBM50374564(CHEMBL255553)
Affinity DataIC50: 2.49E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374567BDBM50374567(CHEMBL269934)
Affinity DataIC50: 2.55E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374569BDBM50374569(CHEMBL271643)
Affinity DataIC50: 2.70E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374575BDBM50374575(CHEMBL403928)
Affinity DataIC50: 2.95E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374562BDBM50374562(CHEMBL402401)
Affinity DataIC50: 3.80E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374570BDBM50374570(CHEMBL402592)
Affinity DataIC50: 4.33E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374573BDBM50374573(CHEMBL260602)
Affinity DataIC50: 4.73E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374576BDBM50374576(CHEMBL402800)
Affinity DataIC50: 4.86E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Inspire Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50374563BDBM50374563(CHEMBL257651)
Affinity DataIC50: 9.90E+3nMAssay Description:Antagonist activity at P2Y12 receptor assessed as platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed