Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50040404
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393706BDBM50393706(CHEMBL2158999)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017712BDBM50017712(Apoplon | 3,4,5-trimethoxybenzoyl methyl reserpate...)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393707BDBM50393707(CHEMBL2158998)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393711BDBM50393711(CHEMBL358518)
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393710BDBM50393710(CHEMBL422481)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393709BDBM50393709(CHEMBL2158996)
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393708BDBM50393708(CHEMBL2158997)
Affinity DataIC50: 1.81E+4nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393714BDBM50393714(CHEMBL142493)
Affinity DataIC50: 2.43E+4nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393713BDBM50393713(CHEMBL2158995)
Affinity DataIC50: 2.65E+4nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393715BDBM50393715(CHEMBL2158994)
Affinity DataIC50: 2.84E+4nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393712BDBM50393712(CHEMBL434066)
Affinity DataIC50: 2.91E+4nMAssay Description:Inhibition of norA-mediated ethidium bromide efflux in methicillin-resistant Staphylococcus aureus SA-1199B by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed