Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50041053
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50451442BDBM50451442(CHEMBL329402)
Affinity DataIC50: 20nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421539BDBM50421539(CHEMBL88731)
Affinity DataIC50: 25nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421548BDBM50421548(CHEMBL87194)
Affinity DataIC50: 25nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403993BDBM50403993(CHEMBL91418)
Affinity DataIC50: 25nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421538BDBM50421538(CHEMBL313070)
Affinity DataIC50: 25nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421542BDBM50421542(CHEMBL88998)
Affinity DataIC50: 25nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421551BDBM50421551(CHEMBL89425)
Affinity DataIC50: 25nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421540BDBM50421540(CHEMBL89818)
Affinity DataIC50: 32nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421544BDBM50421544(CHEMBL89385)
Affinity DataIC50: 32nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403993BDBM50403993(CHEMBL91418)
Affinity DataIC50: 32nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421549BDBM50421549(CHEMBL422773)
Affinity DataIC50: 32nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50451444BDBM50451444(CHEMBL89230)
Affinity DataIC50: 40nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421541BDBM50421541(CHEMBL91436)
Affinity DataIC50: 40nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421541BDBM50421541(CHEMBL91436)
Affinity DataIC50: 50nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421545BDBM50421545(CHEMBL89847)
Affinity DataIC50: 50nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421537BDBM50421537(CHEMBL87066)
Affinity DataIC50: 79nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50451443BDBM50451443(CHEMBL315939)
Affinity DataIC50: 100nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421544BDBM50421544(CHEMBL89385)
Affinity DataIC50: 100nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421548BDBM50421548(CHEMBL87194)
Affinity DataIC50: 100nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421547BDBM50421547(CHEMBL88810)
Affinity DataIC50: 100nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421542BDBM50421542(CHEMBL88998)
Affinity DataIC50: 126nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421545BDBM50421545(CHEMBL89847)
Affinity DataIC50: 126nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421543BDBM50421543(pdCpisodC | CHEMBL419312)
Affinity DataIC50: 126nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50451445BDBM50451445(CHEMBL89640)
Affinity DataIC50: 158nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421543BDBM50421543(pdCpisodC | CHEMBL419312)
Affinity DataIC50: 158nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421549BDBM50421549(CHEMBL422773)
Affinity DataIC50: 158nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421551BDBM50421551(CHEMBL89425)
Affinity DataIC50: 158nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421546BDBM50421546(CHEMBL86890)
Affinity DataIC50: 158nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421546BDBM50421546(CHEMBL86890)
Affinity DataIC50: 200nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421547BDBM50421547(CHEMBL88810)
Affinity DataIC50: 200nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421538BDBM50421538(CHEMBL313070)
Affinity DataIC50: 200nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421536BDBM50421536(CHEMBL89245)
Affinity DataIC50: 200nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421537BDBM50421537(CHEMBL87066)
Affinity DataIC50: 251nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421536BDBM50421536(CHEMBL89245)
Affinity DataIC50: 251nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421540BDBM50421540(CHEMBL89818)
Affinity DataIC50: 316nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421550BDBM50421550(CHEMBL315937)
Affinity DataIC50: 316nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421550BDBM50421550(CHEMBL315937)
Affinity DataIC50: 631nMAssay Description:Binding affinity at serotonin transporter from rat cerebral cortex by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetSubstance-P receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50421539BDBM50421539(CHEMBL88731)
Affinity DataIC50: 1.26E+3nMAssay Description:Binding affinity at human Tachykinin receptor 1 expressed in CHO cells by [3H]-substance P displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed