Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50041798
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415789BDBM50415789(CHEMBL1093773)
Affinity DataIC50: 63.1nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415788BDBM50415788(CHEMBL1093772)
Affinity DataIC50: 63.1nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415790BDBM50415790(GSK-1564023A | CHEMBL1093774 | US10272074, Example...)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415791BDBM50415791(CHEMBL1089404)
Affinity DataIC50: 158nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415793BDBM50415793(CHEMBL1089744)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415794BDBM50415794(GSK-325971A | CHEMBL1093602)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415792BDBM50415792(CHEMBL1089743)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415807BDBM50415807(CHEMBL1090973)
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415808BDBM50415808(CHEMBL1091054)
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415795BDBM50415795(CHEMBL1089745)
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415796BDBM50415796(CHEMBL1089350)
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415806BDBM50415806(CHEMBL1094035)
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415809BDBM50415809(CHEMBL1091439)
Affinity DataIC50: 316nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415810BDBM50415810(CHEMBL1091440 | US10272074, Example 30)
Affinity DataIC50: 316nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415797BDBM50415797(CHEMBL1089692)
Affinity DataIC50: 398nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415798BDBM50415798(CHEMBL1089600)
Affinity DataIC50: 398nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415811BDBM50415811(CHEMBL1093055)
Affinity DataIC50: 501nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415812BDBM50415812(CHEMBL1091066)
Affinity DataIC50: 794nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415799BDBM50415799(CHEMBL1093352)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415794BDBM50415794(GSK-325971A | CHEMBL1093602)
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cells assessed as inhibition of progesterone-induced effec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415790BDBM50415790(GSK-1564023A | CHEMBL1093774 | US10272074, Example...)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of human PDE4B by ATP-luciferace luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415790BDBM50415790(GSK-1564023A | CHEMBL1093774 | US10272074, Example...)
Affinity DataIC50: 3.16E+3nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cells assessed as inhibition of progesterone-induced effec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415794BDBM50415794(GSK-325971A | CHEMBL1093602)
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human PDE4B by ATP-luciferace luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415792BDBM50415792(CHEMBL1089743)
Affinity DataIC50: 5.01E+3nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cells assessed as inhibition of progesterone-induced effec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415813BDBM50415813(CHEMBL1091320)
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415790BDBM50415790(GSK-1564023A | CHEMBL1093774 | US10272074, Example...)
Affinity DataEC50: >6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as renilla luciferase transactivation activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415801BDBM50415801(CHEMBL1093354)
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415796BDBM50415796(CHEMBL1089350)
Affinity DataEC50: >6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as renilla luciferase transactivation activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415802BDBM50415802(CHEMBL1089707)
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415792BDBM50415792(CHEMBL1089743)
Affinity DataEC50: >6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as renilla luciferase transactivation activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415800BDBM50415800(CHEMBL1093353)
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415794BDBM50415794(GSK-325971A | CHEMBL1093602)
Affinity DataEC50: >6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as renilla luciferase transactivation activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415814BDBM50415814(CHEMBL1094032)
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415805BDBM50415805(CHEMBL1094034)
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415803BDBM50415803(CHEMBL1094031)
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415804BDBM50415804(CHEMBL1094033)
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415796BDBM50415796(CHEMBL1089350)
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in african green monkey CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415792BDBM50415792(CHEMBL1089743)
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in african green monkey CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415794BDBM50415794(GSK-325971A | CHEMBL1093602)
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in african green monkey CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415790BDBM50415790(GSK-1564023A | CHEMBL1093774 | US10272074, Example...)
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415796BDBM50415796(CHEMBL1089350)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cells assessed as inhibition of progesterone-induced effec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415794BDBM50415794(GSK-325971A | CHEMBL1093602)
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415796BDBM50415796(CHEMBL1089350)
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415796BDBM50415796(CHEMBL1089350)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in african green monkey CV1 cells assessed as inhibition of aldosterone-induced eff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415792BDBM50415792(CHEMBL1089743)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in african green monkey CV1 cells assessed as inhibition of aldosterone-induced eff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415796BDBM50415796(CHEMBL1089350)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of human PDE4B by ATP-luciferace luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415792BDBM50415792(CHEMBL1089743)
Affinity DataEC50: >2.00E+4nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415792BDBM50415792(CHEMBL1089743)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human PDE4B by ATP-luciferace luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415790BDBM50415790(GSK-1564023A | CHEMBL1093774 | US10272074, Example...)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in african green monkey CV1 cells assessed as inhibition of aldosterone-induced eff...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetMineralocorticoid receptor(Human)
Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50415790BDBM50415790(GSK-1564023A | CHEMBL1093774 | US10272074, Example...)
Affinity DataEC50: >2.00E+4nMAssay Description:Antagonist activity at human mineralocorticoid receptor expressed in african green monkey CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Displayed 1 to 50 (of 51 total ) | Next | Last >>
Jump to: