Compile Data Set for Download or QSAR
Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 50041968
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50080818BDBM50080818((-)-lobeline | 2-(6-(2-Hydroxy-2-phenylethyl)-1-me...)
Affinity DataKi:  2.51nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50080818BDBM50080818((-)-lobeline | 2-(6-(2-Hydroxy-2-phenylethyl)-1-me...)
Affinity DataKi:  5.01nMAssay Description:Displacement of [3H]epibatidine from human nAChR alpha4beta2 receptor expressed in human HEK293T cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82070BDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  12.6nMAssay Description:Displacement of [3H]epibatidine from human nAChR alpha4beta2 receptor expressed in human HEK293T cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419742BDBM50419742(CHEMBL1947055)
Affinity DataKi:  31.6nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419732BDBM50419732(CHEMBL1947053)
Affinity DataKi:  31.6nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419740BDBM50419740(CHEMBL1946189)
Affinity DataKi:  39.8nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419732BDBM50419732(CHEMBL1947053)
Affinity DataKi:  79.4nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419746BDBM50419746(CHEMBL1946188)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419749BDBM50419749(CHEMBL1947058)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419738BDBM50419738(CHEMBL1947206)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419735BDBM50419735(CHEMBL1947059)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419750BDBM50419750(CHEMBL1947060)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419742BDBM50419742(CHEMBL1947055)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419734BDBM50419734(CHEMBL1947056)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419738BDBM50419738(CHEMBL1947206)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419745BDBM50419745(CHEMBL1794606)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82070BDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419739BDBM50419739(CHEMBL1946187)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419733BDBM50419733(CHEMBL1947054)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419737BDBM50419737(CHEMBL1947062)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419734BDBM50419734(CHEMBL1947056)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419740BDBM50419740(CHEMBL1946189)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419736BDBM50419736(CHEMBL1947061)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50080818BDBM50080818((-)-lobeline | 2-(6-(2-Hydroxy-2-phenylethyl)-1-me...)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419730BDBM50419730(CHEMBL1947049)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419736BDBM50419736(CHEMBL1947061)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419748BDBM50419748(CHEMBL1947057)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419749BDBM50419749(CHEMBL1947058)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419750BDBM50419750(CHEMBL1947060)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419739BDBM50419739(CHEMBL1946187)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82070BDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]MLA from nAChR alpha7 receptor in human SH-SY5Y cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419733BDBM50419733(CHEMBL1947054)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419739BDBM50419739(CHEMBL1946187)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]MLA from nAChR alpha7 receptor in human SH-SY5Y cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419744BDBM50419744(CHEMBL1946185)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419748BDBM50419748(CHEMBL1947057)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419740BDBM50419740(CHEMBL1946189)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]MLA from nAChR alpha7 receptor in human SH-SY5Y cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419731BDBM50419731(CHEMBL1947051)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419741BDBM50419741(CHEMBL1947048)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419751BDBM50419751(DEPTROPINE)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419753BDBM50419753(CHEMBL1947047)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419743BDBM50419743(CHEMBL1947205)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419735BDBM50419735(CHEMBL1947059)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82070BDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419730BDBM50419730(CHEMBL1947049)
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [3H]MLA from nAChR alpha7 receptor in human SH-SY5Y cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419731BDBM50419731(CHEMBL1947051)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419730BDBM50419730(CHEMBL1947049)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419733BDBM50419733(CHEMBL1947054)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]MLA from nAChR alpha7 receptor in human SH-SY5Y cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetSoluble acetylcholine receptor(California sea hare)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419751BDBM50419751(DEPTROPINE)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAcetylcholine-binding protein(Great pond snail)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419747BDBM50419747(CHEMBL1947052)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis acetylcholine binding protein expressed using baculoviral system after 1.5 hrs by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50419742BDBM50419742(CHEMBL1947055)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H]MLA from nAChR alpha7 receptor in human SH-SY5Y cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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