Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50042216
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422267BDBM50422267(CHEMBL263079)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422250BDBM50422250(CHEMBL268174)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422234BDBM50422234(CHEMBL6412)
Affinity DataIC50: 10nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422254BDBM50422254(CHEMBL6785)
Affinity DataIC50: 13nMAssay Description:Inhibition of specific binding of [125-I] ET-1 to human Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422257BDBM50422257(CHEMBL6555)
Affinity DataIC50: 16nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50034435BDBM50034435(BMS-182874 | 5-Dimethylamino-naphthalene-1-sulfoni...)
Affinity DataIC50: 50nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422248BDBM50422248(CHEMBL6800)
Affinity DataIC50: 63nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422244BDBM50422244(CHEMBL268339)
Affinity DataIC50: 126nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422246BDBM50422246(CHEMBL6553)
Affinity DataIC50: 158nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422264BDBM50422264(CHEMBL6761)
Affinity DataIC50: 200nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422249BDBM50422249(CHEMBL266277)
Affinity DataIC50: 251nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422243BDBM50422243(CHEMBL6297)
Affinity DataIC50: 251nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422233BDBM50422233(CHEMBL6624)
Affinity DataIC50: 316nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422265BDBM50422265(CHEMBL268116)
Affinity DataIC50: 316nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422241BDBM50422241(CHEMBL415106)
Affinity DataIC50: 398nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422245BDBM50422245(CHEMBL6588)
Affinity DataIC50: 501nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422266BDBM50422266(CHEMBL7019)
Affinity DataIC50: 631nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422263BDBM50422263(CHEMBL6382)
Affinity DataIC50: 631nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422258BDBM50422258(CHEMBL6399)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422253BDBM50422253(CHEMBL6583)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422261BDBM50422261(CHEMBL415292)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422236BDBM50422236(CHEMBL6463)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422256BDBM50422256(CHEMBL268387)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422240BDBM50422240(CHEMBL6411)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422262BDBM50422262(CHEMBL6433)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422255BDBM50422255(CHEMBL6630)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422237BDBM50422237(CHEMBL266315)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422238BDBM50422238(CHEMBL6576)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422247BDBM50422247(CHEMBL6543)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422242BDBM50422242(CHEMBL6400)
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422232BDBM50422232(CHEMBL269237)
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422251BDBM50422251(CHEMBL6660)
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422235BDBM50422235(CHEMBL6647)
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422259BDBM50422259(CHEMBL266684)
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422239BDBM50422239(CHEMBL6468)
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422252BDBM50422252(CHEMBL6778)
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422260BDBM50422260(CHEMBL6566)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of specific binding of [125-I]ET-1 to human endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article
PubMed