Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50043063
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435322BDBM50435322(CHEMBL2391376)
Affinity DataIC50: 180nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435311BDBM50435311(CHEMBL2391351)
Affinity DataIC50: 210nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435312BDBM50435312(CHEMBL2391354)
Affinity DataIC50: 270nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435314BDBM50435314(CHEMBL2391352)
Affinity DataIC50: 390nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435329BDBM50435329(CHEMBL2391368)
Affinity DataIC50: 430nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435316BDBM50435316(CHEMBL2391382)
Affinity DataIC50: 500nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435340BDBM50435340(CHEMBL2391358)
Affinity DataIC50: 590nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435319BDBM50435319(CHEMBL2391379)
Affinity DataIC50: 930nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435339BDBM50435339(CHEMBL2391359)
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435313BDBM50435313(CHEMBL2391353)
Affinity DataIC50: 2.25E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435341BDBM50435341(CHEMBL2391357)
Affinity DataIC50: 3.25E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435328BDBM50435328(CHEMBL2391369)
Affinity DataIC50: 7.24E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435336BDBM50435336(CHEMBL2391362)
Affinity DataIC50: 7.60E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435324BDBM50435324(CHEMBL2391374)
Affinity DataIC50: 8.41E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435335BDBM50435335(CHEMBL2391363)
Affinity DataIC50: 8.83E+3nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435333BDBM50435333(CHEMBL2391365)
Affinity DataIC50: 1.15E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435315BDBM50435315(CHEMBL2391539)
Affinity DataIC50: 1.16E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435320BDBM50435320(CHEMBL2391378)
Affinity DataIC50: 1.18E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435318BDBM50435318(CHEMBL2391380)
Affinity DataIC50: 1.52E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435337BDBM50435337(CHEMBL2391361)
Affinity DataIC50: 1.52E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435325BDBM50435325(CHEMBL2391373)
Affinity DataIC50: 1.58E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435334BDBM50435334(CHEMBL2391364)
Affinity DataIC50: 1.63E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435317BDBM50435317(CHEMBL2391381)
Affinity DataIC50: 1.80E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435327BDBM50435327(CHEMBL2391371)
Affinity DataIC50: 1.88E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435323BDBM50435323(CHEMBL2391375)
Affinity DataIC50: 2.11E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435343BDBM50435343(ESAPRAZOLE)
Affinity DataIC50: 2.72E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435326BDBM50435326(CHEMBL2391372)
Affinity DataIC50: 8.68E+4nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435338BDBM50435338(CHEMBL2391360)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435321BDBM50435321(CHEMBL2391377)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435342BDBM50435342(CHEMBL2391356)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435332BDBM50435332(CHEMBL2391366)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435331BDBM50435331(CHEMBL2391367)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Nensius Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435330BDBM50435330(CHEMBL2391540)
Affinity DataIC50: 1.00E+5nMAssay Description:Binding affinity to sigma1 receptor (unknown origin) by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed