Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50043202
TargetVitamin D3 receptor(Human)
Teikyo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50437338BDBM50437338(CHEMBL2407821)
Affinity DataEC50:  0.0100nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Teikyo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50200182BDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.0260nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Teikyo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50437335BDBM50437335(CHEMBL2407824)
Affinity DataEC50:  0.0440nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Teikyo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50437336BDBM50437336(CHEMBL2407823)
Affinity DataEC50:  0.150nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Teikyo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50437334BDBM50437334(CHEMBL2407825)
Affinity DataEC50:  0.210nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Teikyo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50437337BDBM50437337(CHEMBL2407822)
Affinity DataEC50:  0.290nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Teikyo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50437333BDBM50437333(CHEMBL2407826)
Affinity DataEC50:  0.680nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed