Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50043412
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440788BDBM50440788(CHEMBL2431249)
Affinity DataKi:  0.0170nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440782BDBM50440782(CHEMBL2431246)
Affinity DataKi:  0.0190nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356282BDBM50356282(CHEMBL1910936)
Affinity DataKi:  0.0210nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440784BDBM50440784(CHEMBL2431253)
Affinity DataKi:  0.0210nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440791BDBM50440791(CHEMBL2431256)
Affinity DataKi:  0.0220nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440793BDBM50440793(CHEMBL2431254)
Affinity DataKi:  0.0340nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50385314BDBM50385314(CHEMBL2035981)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440786BDBM50440786(CHEMBL2431251)
Affinity DataKi:  0.0450nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440789BDBM50440789(CHEMBL2431248)
Affinity DataKi:  0.0460nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440790BDBM50440790(CHEMBL2431247)
Affinity DataKi:  0.0560nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440785BDBM50440785(CHEMBL2431252)
Affinity DataKi:  0.0940nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440789BDBM50440789(CHEMBL2431248)
Affinity DataIC50: 0.0970nMAssay Description:Antagonist activity at CGRP receptor (unknown origin) by cell based cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440792BDBM50440792(CHEMBL2431255)
Affinity DataKi:  0.110nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440783BDBM50440783(CHEMBL2429882)
Affinity DataKi:  0.110nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440789BDBM50440789(CHEMBL2431248)
Affinity DataIC50: 0.390nMAssay Description:Antagonist activity at CGRP receptor (unknown origin) by cell based cAMP assay in presence of human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50440787BDBM50440787(CHEMBL2431250)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetCalcitonin gene-related peptide type 1 receptor(Human)
Merck Research Labortories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50224431BDBM50224431(N-[(3R,6S)-6-(2,3-difluorophenyl)-2-oxo-1-(2,2,2-t...)
Affinity DataKi:  0.770nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed